MURINEDDU, Gabriele
 Distribuzione geografica
Continente #
NA - Nord America 2.653
EU - Europa 1.484
AS - Asia 763
OC - Oceania 13
Continente sconosciuto - Info sul continente non disponibili 9
SA - Sud America 8
AF - Africa 6
AN - Antartide 1
Totale 4.937
Nazione #
US - Stati Uniti d'America 2.640
UA - Ucraina 673
CN - Cina 639
DE - Germania 233
IT - Italia 169
SE - Svezia 137
FI - Finlandia 107
TR - Turchia 79
GB - Regno Unito 54
FR - Francia 43
BE - Belgio 30
KR - Corea 15
AU - Australia 12
CA - Canada 11
EU - Europa 8
IN - India 8
IR - Iran 8
RO - Romania 7
CZ - Repubblica Ceca 6
BR - Brasile 5
ES - Italia 4
EG - Egitto 3
JP - Giappone 3
SG - Singapore 3
BG - Bulgaria 2
DK - Danimarca 2
HU - Ungheria 2
IQ - Iraq 2
NL - Olanda 2
PT - Portogallo 2
SK - Slovacchia (Repubblica Slovacca) 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AE - Emirati Arabi Uniti 1
AL - Albania 1
AM - Armenia 1
AT - Austria 1
BD - Bangladesh 1
BO - Bolivia 1
CH - Svizzera 1
CL - Cile 1
DZ - Algeria 1
GS - Georgia del Sud e Isole Sandwich Australi 1
IL - Israele 1
JM - Giamaica 1
MC - Monaco 1
MD - Moldavia 1
NG - Nigeria 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PE - Perù 1
PL - Polonia 1
RS - Serbia 1
RU - Federazione Russa 1
SA - Arabia Saudita 1
TH - Thailandia 1
VG - Isole Vergini Britanniche 1
ZA - Sudafrica 1
Totale 4.937
Città #
Chandler 675
Jacksonville 417
Princeton 238
Dearborn 216
Nanjing 192
Ann Arbor 109
Wilmington 105
New York 81
Izmir 76
Sassari 61
Ashburn 58
Nanchang 56
Shenyang 56
Beijing 52
Woodbridge 46
Hebei 43
Changsha 38
Brussels 29
Jiaxing 29
Tianjin 29
Kunming 22
Boardman 21
Andover 19
Ningbo 19
Jinan 17
San Mateo 17
Hangzhou 16
Mountain View 16
Norwalk 16
Seoul 15
Guangzhou 14
San Francisco 13
Helsinki 12
Taizhou 12
Monmouth Junction 11
Zhengzhou 11
Augusta 9
Toronto 9
Auburn Hills 8
Lanzhou 8
Albissola Marina 7
Leawood 7
Rome 7
Edinburgh 6
Los Angeles 6
Quartu Sant'Elena 6
Brno 5
Hanover 5
Horia 5
London 5
Melbourne 5
Ardabil 4
Changchun 4
Frankfurt am Main 4
Houston 4
São Paulo 4
Alghero 3
Haikou 3
Paris 3
Tokyo 3
Aversa 2
Bariano 2
Budapest 2
Canberra 2
Castel Gandolfo 2
Dallas 2
Fuzhou 2
Genoa 2
Hefei 2
Huskvarna 2
Incisa 2
Media 2
Montreal 2
Mumbai 2
Nutley 2
Palermo 2
Quartucciu 2
Seattle 2
Sofia 2
Aarau 1
Abuja 1
Algiers 1
Amsterdam 1
Atlanta 1
Baghdad 1
Bangalore 1
Bangkok 1
Baotou 1
Belgrade 1
Berlin 1
Bologna 1
Bratislava 1
Brierley Hill 1
Cagliari 1
Chengdu 1
Chisinau 1
Cleveland 1
Cochabamba 1
Dolianova 1
Dubai 1
Totale 3.046
Nome #
Thienocinnolinone alkanoic acid derivatives as aldose reductase inhibitors 79
Tricyclic Pyrazoles. Part 8. Synthesis, Biological Evaluation and Modelling of Tricyclic Pyrazole Carboxamides as Potential CB2 Receptor Ligands with Antagonist/Inverse Agonist Properties. 78
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2 ',4 '-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyra zole-3-carboxamide 68
Chiral pyridine N-oxides useful ligands for asymmetric catalysis 67
Synthesis and D2-like binding affinity of new derivatives of N-(1-ethyl-2-pyrrolidinylmethyl)-4,5-dihydro-1H-benzo[g]indole-3-carboxamide and related 4H-[1]Benzothiopyrano[4,3-b]pyrrole and 5,6-Dihydro-4H benzo[6,7]cyclohepta[b]pyrrole-3-carboxamide Analogues 65
Chromophore-modified bis-benzo[g]indazole carboxamides: synthesis and antiproliferactive activity of bis-benzo[g]indazole carboxamides and related dimers 65
Approcci terapeutici contro il cancro. Tradizione e innovazione. 64
Pyridazine N-Oxides. III. Synthesis and “in vitro” antimicrobial properties of N-Oxide derivatives based on tricyclic indeno[2,1-c]pyridazine and benzo [f]cinnoline systems 63
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists 63
Preparation of thieno[3,2-h]cinnolinones as matrix metalloproteinase inhibitors 63
The organic chemistry of drug design and drug action 62
Synthesis and Antineoplastic Evaluation of Novel Unsymmetrical 1,3,4-Oxadiazoles 60
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism 60
Chemistry of tricyclic-based heterocycles as useful scaffolds for phosphodiesterase 10A ligands 59
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands 59
A critical review of both the synthesis approach and the receptor profile of the 8-chloro-1-(2′,4′-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6- tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide and analogue derivatives. 59
Correction to Synthesis and antineoplastic evaluation of novel unsymmetrical 1,3,4-oxadiazoles 59
Design of novel 3,6-diazabicyclo[3.1.1]heptane derivatives with potent and selective affinities for α4β2 neuronal nicotinic acetylcholine receptors 57
Composti farmaceutici 56
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors 56
New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking 55
Synthesis, Modelling, and Antimitotic Properties of Tricyclic Systems Characterised by a 2-(5-Phenyl-1H-pyrrol-3-yl)-1,3,4-oxadiazole Moiety 55
An overview on different classes of viral entry and respiratory syncitial virus (RSV) fusion inhibitors 54
Synthesis and cytotoxicity of novel hexahydrothienocyclohepta-pyridazinone derivatives 53
CAPITOLO 41. Antielmintici 53
Pyrazole derivatives having affinity for CB1 and/or CB2 receptors 52
Design, Synthesis and preliminary biological data of new ligands for neuronal nicotinic acetylcholine receptors 51
Synthesis and cytotoxicity evaluation of thiophene analogues of 1-methyl-2,3-bis(hydroxymethyl)benzo[g]indole bis[N-(2-propyl)carbamate] 50
Tricyclic pyrazole derivatives as cannabinoid receptor antagonist 50
Ossadiazoli ad attività antiproliferativa 50
Development and characterization of novel cannabinoid derivatives based on diarylpyridazine scaffold. 50
Preliminary anti-coxsackie activity of novel 1-[4-(5,6-dimethyl(h)1h(2h)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas 49
I 3,6-diazabiciclo[3.1.1]eptani: una nuova serie di potenti agonisti per i recettori μ degli oppioidi 48
Oxadiazoles having anti proliferative activity 48
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands 48
Design of a new class of chiral C2-symmetric dipyridylmethane ligands and their application in asymmetric catalysis 48
Novel diazabicycloalkane delta opioid agonists 47
Oxadiazoles having antiproliferative activity 46
Manuale di chimica farmaceutica. Progettazione, meccanismo d'azione e metabolismo dei farmaci 46
Pharmaceutical Compounds 46
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS 46
Synthesis and anti-HIV-1 activity of new delavirdine analogues carrying arylpyrrole moieties 46
Synthesis of biologically active bridged diazabicycloheptanes 45
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzolglindazole-based ligands for cannabinoid receptors 45
Synthesis, modelling, and m-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes 44
Tricyclic pyrazoles Part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands 44
Synthesis and biological evaluation of novel CB2 ligands 44
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors 44
Pharmaceutical compounds 44
Synthesis and cytotoxicity of substituted 2-benzylnaphth[2,3-d]imidazoles 44
Synthesis and μ-opioid receptor affinity of fused .bicyclic analogues of N-3(9)-Arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes (DBNs) 43
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands 43
Synthesis and pharmacological evaluation of novel 4-Alkyl-5-thien-2'-yl pyrazole carboxamides 42
3-{2-[Bis-(4-fluorophenyl)methoxy]ethyl}-6-substituted-3,6-diazabicyclo[ 3.1.1]heptanes as novel potent dopamine uptake inhibitors 42
3-(5-Phenyl[1,3,4]oxadiazol-2-yl)-1H-benzo]g]indole and related compounds: synthesis and cytotoxic acitivities 42
Pharmaceutical compounds 42
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation 42
Ring-fused pyrazole derivates as ligands for cannabinoid receptors: synthesis and investigation of structure-activity relationships 41
Synthesis and cytotoxic activities of pyrrole[2,3-d]pyridazin-4-one derivatives 41
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonists 41
Tricyclic pyrazoles. Part 3. Synthesis, biological evaluation and molecular modelling of analogues of the cannabinoid antagonist NESS 0327 41
Pharmaceutical compounds 40
5,6-Dichloro-2-phenyl-benzotriazoles: New potent inhibitors of orthohantavirus 40
Sintesi di 1,10-fenantroline chirali a simmetria C2 derivati da monoterpeni naturali quali utili leganti per la catalisi asimmetrica 40
RNA-viruses. Enzymatic and receptorial inhibitors. Research signpost keral, India, (RNA-viruses. Enzymatic and recptoral inhibitors. 39
N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as μ-opioid receptor agonists. Effects on μ-affinity of arylalkenyl chain modifications 39
Synthesis and analgesic-antiinflammatory activities of novel acylarylhydrazones with a 5-phenyl-4-R-3-pyrrolyl-acyl moiety 39
Tricyciclic Pyrazoles. Synthesis and bilogical evaluation of novel 4,5-dihydro-1H-6-oxa-cicloepta[1,2-c]pyrazole-based analogues of cannabinoid antagonist NESS-0327 39
Synthesis and μ-opioid receptor affinity of heteroaromatic analogues of N-3(9)-Arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes (DBNs) 39
Synthesis and tumor cell lines inhibition of 1,3,4.oxadiazoles linked to tricyclic pyrroles 39
Different classes of CB2 Ligands Potentially Useful in the Treatment of Pain. 38
Synthesis of chiral C2-symmetric 1,10-phenanthrolines from naturally occurring monoterpenes 38
Sintesi di nuovi diazatriciclodicani (DTDs). Effetto della variazione strutturale della catena cinnamilica sulla μ-affinità e sull’analgesia oppioide 38
Pharmaceutical compounds 38
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. . 38
NESS06SM reduces body weight with an improved profile relative to SR141716A 37
Pharmaceutical compounds 36
Synthesis and application in asymmetric copper(I)-catalyzed allylic oxidation of a new chiral 1,10-phenantroline derived from pinene 36
Substituted 3,8-diazabicyclo[3.2.1]octane compounds 36
Sintesi di nuovi leganti chirali dipiridilmetanici e loro applicazione nella sostituzione allilica palladio-catalizzata 35
Versatility of the pyridazine system: chemistry and biology 35
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors 35
Myrtanil substituent in 3 position of pirazole ring determines CB1 agonism of novel 4,5-dihydrobenzo-oxa-cycloheptapyrazole cannabinoids 34
Oxadiazoles having antiproliferative activity 34
Diazacyclic compounds having affinity for opioid receptors 34
Synthesis and cytotoxic activities of 3-(5-phenyl-[1.3.4]oxadiazol-2-yl)-1H-benzo[g]indole and related compounds 34
I farmaci antivirali. Dalla progettazione all’impiego terapeutico. 34
Chimica farmaceutica. Con e-book 33
Synthesis, Pharmacological Evaluation and Docking Studies of Pyrrole Structure-Based CB2 Receptor Antagonists 33
Sintesi e affinità per i recettori oppioidi di nuovi N3-propionil-N6-naftilprop(en)il-3,6-diazabiciclo[3.3.1]eptani 33
Pharmaceutical compounds 32
Pharmaceutical Compounds 32
Chimica farmaceutica 32
Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties 32
Principi generali. In: Chimica Tossicologica 31
Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazoles: A versatile architecture for CB2 selective ligands 31
Tricyclic thieno-pyrazoles as new potent and selective CB2 ligands 31
Pyrazolo-naphthyridines: Design and Synthesis of potential CB-ligands 30
A survey of Recent Patents on CB2 Agonists in the Management of Pain 30
New tricyclic pyrazole derivatives as CB1 antagonists having improved activity towards food intake and weight control 29
Totale 4.540
Categoria #
all - tutte 20.875
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 20.875


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019195 0 0 0 0 0 0 0 0 0 0 9 186
2019/20201.231 315 3 106 7 103 188 218 15 126 38 109 3
2020/2021920 110 5 138 12 111 32 124 23 128 135 82 20
2021/2022572 67 6 9 7 8 5 28 48 51 37 61 245
2022/20231.271 130 78 27 229 110 210 2 161 228 8 56 32
2023/2024305 58 26 15 7 37 81 1 55 3 4 18 0
Totale 5.037