Sfoglia per Autore
Synthesis and Pharmacological Evaluation of 1,2-Diphenyl-4-(aminomethyl)imidazoles with Clozapine-Like Mixed Activities at Dopamine D2, Serotonin, and GABAA Receptors. XXI° Congresso Nazionale della Società Chimica Italiana, Torino, 22-27 Giugno 2003, FA-CO-001 (Atti, Vol.1; Conferenze Plenarie-Comunicazioni Orali)
2003-01-01 Asproni, Battistina; A., Pau; R., Cerri; L., Dazzi; E., Maciocco; E., Sanna; C., Altomare; G., Trapani; G., Biggio
Nuovi Derivati 1,2-difenil-imidazolici come potenti ed efficaci modulatori allosterici positivi del recettore GABAA. Sardinia Chem 2004. Giornata di studio dedicata alla chimica organica delle molecole biologicamente attive. P32 (pag. 95)
2004-01-01 Asproni, Battistina; A., Pau; R., Cerri; M. P., Mascia; E., Sanna; G., Biggio
Nuovi derivati 1,2-difenil-imidazolici come potenti ed efficaci modulatori allosterici positivi del recettore GABAA
2004-01-01 Asproni, Battistina; Pau, Amedeo; Cerri, Riccardo; Mascia, Maria Paola; Biggio, Giovanni; Sanna, Enrico
Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives
2004-01-01 Pau, Amedeo; Asproni, Battistina; Boatto, Gianpiero; Grella, Giuseppe Enrico; De Caprariis, P.; Costantino, L.; Pinna, Gerard Aime
Determination amphetamine-derived designer drugs in human urine by SPE extraction and capillary electrophoresis with mass spectrometry detection
2005-01-01 Boatto, Gianpiero; Nieddu, M; Carta, Antonio; Pau, ; Palomba, M; Asproni, Battistina; Cerri, R.
Synthesis, Structure-Activity Relationships at the GABAA Receptor in Rat Brain, and Differential Electrophysiological Profile at the Recombinant Human GABAA Receptor of a Series of Substituted 1,2-Diphenylimidazoles
2005-01-01 Asproni, Battistina; Talani, G; Busonero, F; Pau, A; Sanna, S; Cerri, R; Mascia, M. P.; Sanna, E; Biggio, G.
Synthesis and structure-activity relationships at GABAA receptor in rat brain and differential electrophysiological profile at recombinant human GABAA receptor of a series of substituted 1,2-diphenyl-imidazoles
2005-01-01 Asproni, B.; Talani, G.; Busonero, F.; Pau, Amedeo; Sanna, E.; Cerri, R.; Mascia, M. P.; Sanna, E.; Biggio, AND G.
Ethyl 2-(4-bromophenyl)-1-(2,4-dichlorophenyl)-1H-4-imidazolecarboxylate is a Novel Positive Modulator of GABAA Receptors
2005-01-01 Mascia, M. P.; Asproni, Battistina; Busonero, F; Talani, G; Maciocco, E; Pau, Amedeo; Cerri, R; Sanna, E; Biggio, G.
Thienocinnolinone alkanoic acid derivatives as aldose reductase inhibitors
2006-01-01 Pau, Amedeo; Asproni, Battistina; Murineddu, Gabriele; Boatto, Gianpiero; Grella, Giuseppe Enrico; Rakowitz, D.; Costantino, L.; Pinna, Gerard Aime
Synthesis and SAR study of 2-substituted imidazo[2,1-b][1,3]benzothiazoles and related compounds endowed with affinity for dopamine D2 receptors as potential antipsychotics
2008-01-01 Asproni, Battistina; Kehler, J.; S., Simula; G., Porcu
Synthesis and sar study of 2-substituted imidazo[2,1-b] [1,3]benzothiazoles and related compounds endowed with affinity for dopamine D2receptors as potential antipsychotics
2008-01-01 Asproni, Battistina; Kehler, Jan; Mura, Stefania; Porcu, Giovanna; Simula, Sergio
Synthesis and cytotoxicity of novel hexahydrothienocyclohepta-pyridazinone derivatives
2009-01-01 Pau, Amedeo; Murineddu, Gabriele; Asproni, Battistina; Murruzzu, C; Grella, Giuseppe Enrico; Pinna, Gerard Aime; Curzu, Maria Michela; Marchesi, I; Bagella, Luigi Marco
Ring-fused pyrazole derivates as ligands for cannabinoid receptors: synthesis and investigation of structure-activity relationships
2011-01-01 Deligia, F; Dore, A; Pinna, Giansalvo; Asproni, B; Murineddu, Gabriele; Pinna, Gerard Aime
Synthesis and SAR study of new phenylimidazole-pyrazolo[1,5-c]quinazolines as potent phosphodiesterase 10A inhibitors
2011-01-01 Asproni, Battistina; Murineddu, Gabriele; Pau, Amedeo; Pinna, Gerard Aime; Langgard, M; Christoffersen, C. T.; Nielsen, J; Kehler, J.
Synthesis of biologically active bridged diazabicycloheptanes
2012-01-01 Murineddu, Gabriele; Asproni, Battistina; Curzu, Maria Michela; Pinna, G; Dore, A; Pau, Amedeo; Deligia, F; Pinna, Gerard Aime
Tricyclic pyrazoles. Part 5. novel 1,4-Dihydroindeno[1,2-c]pyrazole CB2 ligands using molecular hybridization based on scaffold hopping
2012-01-01 Murineddu, Gabriele; Asproni, Battistina; Ruiu, S; Deligia, F; Falzoi, M; Pau, Amedeo; Thomas, Bf; Zhang, Y; Pinna, Gerard Aime; Pani, L; Lazzari, P.
Synthesis and pharmacological evaluation of novel 4-Alkyl-5-thien-2'-yl pyrazole carboxamides
2012-01-01 Lazzari, P; Pau, Amedeo; Tambaro, S; Asproni, Battistina; Ruiu, S; Pinna, G; Mastinu, A; Curzu, Maria Michela; Reali, R; Bottazzi, Me; Pinna, Gerard Aime; Murineddu, Gabriele
A survey of Recent Patents on CB2 Agonists in the Management of Pain
2012-01-01 Murineddu, Gabriele; Asproni, Battistina; Pinna, Gerard Aime
Different classes of CB2 Ligands Potentially Useful in the Treatment of Pain.
2013-01-01 Murineddu, Gabriele; Deligia, F; Dore, A; Pinna, Gerard Aime; Asproni, Battistina; Pinn, Ga
Synthesis and biological evaluation of novel delta (δ) opioid receptor ligands with diazatricyclodecane skeletons
2013-01-01 Loriga, G; Lazzari, P; Ruiu, S; Marchese, G; Manca, I; Casu, G. L.; Dessì, C; Pinna, Gerard Aime; Asproni, Battistina; Murineddu, Gabriele
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