Sfoglia per Autore
Quinoline tricyclic derivatives. Design, synthesis and evaluation of the antiviral activity of three new classes of RNA-Dependent RNA Polymerase inhibitors
2011-01-01 Carta, Antonio; Briguglio, Irene; Piras, Sandra; Corona, Paola; Boatto, Gianpiero; M., Nieddu; Giunchedi, Paolo; M. E., Marongiu; G., Giliberti; F., Iuliano; S., Blois; C., Ibba; B., Busonera; P., La Colla
Inhibition of RNA helicases of ssRNA+virus belonging toFlaviviridae,CoronaviridaeandPicornaviridaefamilies
2011-01-01 Piras, Sandra; Corona, Paola; Carta, Antonio; Briguglio, Irene
5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4.
2012-01-01 Vitale, Gabriella; Corona, Paola; Loriga, M; Carta, Antonio; Paglietti, G; Giliberti, G; Sanna, G; Farci, P; Marongiu, Me; La Colla, P.
Structure-based selectivity optimization of piperidine-pteridine derivatives as potent Leishmania pteridine reductase inhibitors
2012-01-01 Corona, Paola; Gibellini, F; Cavalli, A; Saxena, P; Carta, Antonio; Loriga, M; Luciani, R; Paglietti, G; Guerrieri, D; Nerini, E; Gupta, S; Hannaert, V; Michels, Pam; Ferrari, S; Costi, Pm
SAR and Anti-Mycobacterial Activity of Quinolones and Triazoloquinolones: An Update
2013-01-01 Briguglio, Irene; Piras, Sandra; Corona, Paola; Pirisi, Maria Antonietta; Jabes, D; Carta, Antonio
2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7trifluoromethylquinoxalines as anticancer agents Inhibitors of folate enzymes
2014-01-01 Piras, Sandra; Carta, Antonio; Briguglio, Irene; Corona, Paola; Paglietti, Giuseppe; Luciani, R; Costi, M. P; Steania Ferrari, S.
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines
2014-01-01 Loddo, R; Briguglio, Irene; Corona, Paola; Piras, Sandra; Loriga, M; Paglietti, G; Carta, Antonio; Sanna, G; Giliberti, G; Ibba, C; Farci, P; La Colla, P.
Benzotriazole: an overview on its versatile biological behaviour
2015-01-01 Briguglio, Irene; Piras, Sandra; Corona, Paola; Gavini, Elisabetta; Nieddu, M; Boatto, Gianpiero; Carta, Antonio
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives
2015-01-01 Briguglio, Irene; Loddo, Roberta; Laurini, Erik; Fermeglia, Maurizio; Piras, Sandra; Corona, Paola; Giunchedi, Paolo; Gavini, Elisabetta; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; La Colla, Paolo; Pricl, Sabrina; Carta, Antonio
A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems
2016-01-01 Carta, Antonio; Briguglio, Irene; Piras, Sandra; Corona, Paola; Ibba, R.; Laurini, E.; Fermeglia, M.; Pricl, S.; Desideri, N.; Atzori, E. M.; La Colla, P.; Collu, G.; Delogu, I.; Loddo, R.
Synthesis of 2-(Quinoxalin-2-ylamino-benzotriazolyl) Pentanedioic Derivatives as Potential Anti-Folate Agents
2016-01-01 Briguglio, Irene; Piras, Sandra; Corona, Paola; Pirisi, Maria Antonietta; Burrai, L; Boatto, Gianpiero; Gavini, Elisabetta; Rassu, Giovanna
Triazolopyridinyl-acrylonitrile derivatives as antimicrotubule agents: synthesis, in vitro and in silico characterization of antiproliferative activity, inhibition of tubulin polymerization and binding thermodynamics
2017-01-01 Briguglio, Irene; Laurini, Erik; Pirisi, Maria Antonietta; Piras, Sandra; Corona, Paola; Fermeglia, Maurizio; Pricl, Sabrina; Carta, Antonio
Antiviral activities of 5-chlorobenzotriazole derivatives
2018-01-01 Ibba, Roberta; Corona, P; Carta, A; Giunchedi, P; Loddo, R; Sanna, Giuseppina; Delogu, Ilenia; Piras, S
Quinoxaline derivatives as new inhibitors of coxsackievirus B5
2018-01-01 Carta, Antonio; Giuseppina, Sanna; Briguglio, Irene; Madeddu, Silvia; Vitale, Gabriella; Piras, Sandra; Corona, Paola; Peana, Alessandra Tiziana; Laurini, Erik; Fermeglia, Maurizio; Pricl, Sabrina; Alessandra, Serra; Carta, Elisa; Loddo, Roberta; Giliberti, Gabriele
Enhancement of antimicrobial activity of pump inhibitors associating drugs
2019-01-01 Usai, Donatella; Donadu, Matthew; Bua, Alessandra; Molicotti, Paola; Zanetti, Stefania; Piras, Sandra; Corona, Paola; Ibba, Roberta; Carta, Antonio
Design, synthesis and antitubercular activity of 4-alkoxy-triazoloquinolones able to inhibit the M. tuberculosis DNA gyrase
2019-01-01 Carta, Antonio; Bua, Alessandra; Corona, Paola; Piras, Sandra; Briguglio, Irene; Molicotti, Paola; Zanetti, Stefania; Laurini, Erik; Aulic, Suzana; Fermeglia, Maurizio; Pricl, Sabrina
Poly (ethyl 2-cyanoacrylate) nanoparticles (PECA-NPs) as possible agents in tumor treatment
2019-01-01 Obinu, Antonella; Rassu, Giovanna; Corona, Paola; Maestri, Marcello; Riva, Federica; Miele, Dalila; Giunchedi, Paolo; Gavini, Elisabetta
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands
2019-01-01 Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A.
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors
2019-01-01 Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A.
Dichloro-phenyl -benzotriazoles: a new selective class of human respiratory syncytial virus entry inhibitors
2019-01-01 Piras, Sandra; Sanna, Giuseppina; Carta, Antonio; Corona, Paola; Ibba, Roberta; Loddo, Roberta; Madeddu, Silvia; Caria, Paola; Aulic, Suzana; Laurini, Erik; Fermeglia, Maurizio; Pricl, Sabrina
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Quinoline tricyclic derivatives. Design, synthesis and evaluation of the antiviral activity of three new classes of RNA-Dependent RNA Polymerase inhibitors | 1-gen-2011 | Carta, Antonio; Briguglio, Irene; Piras, Sandra; Corona, Paola; Boatto, Gianpiero; M., Nieddu; Giunchedi, Paolo; M. E., Marongiu; G., Giliberti; F., Iuliano; S., Blois; C., Ibba; B., Busonera; P., La Colla | |
Inhibition of RNA helicases of ssRNA+virus belonging toFlaviviridae,CoronaviridaeandPicornaviridaefamilies | 1-gen-2011 | Piras, Sandra; Corona, Paola; Carta, Antonio; Briguglio, Irene | |
5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4. | 1-gen-2012 | Vitale, Gabriella; Corona, Paola; Loriga, M; Carta, Antonio; Paglietti, G; Giliberti, G; Sanna, G; Farci, P; Marongiu, Me; La Colla, P. | |
Structure-based selectivity optimization of piperidine-pteridine derivatives as potent Leishmania pteridine reductase inhibitors | 1-gen-2012 | Corona, Paola; Gibellini, F; Cavalli, A; Saxena, P; Carta, Antonio; Loriga, M; Luciani, R; Paglietti, G; Guerrieri, D; Nerini, E; Gupta, S; Hannaert, V; Michels, Pam; Ferrari, S; Costi, Pm | |
SAR and Anti-Mycobacterial Activity of Quinolones and Triazoloquinolones: An Update | 1-gen-2013 | Briguglio, Irene; Piras, Sandra; Corona, Paola; Pirisi, Maria Antonietta; Jabes, D; Carta, Antonio | |
2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7trifluoromethylquinoxalines as anticancer agents Inhibitors of folate enzymes | 1-gen-2014 | Piras, Sandra; Carta, Antonio; Briguglio, Irene; Corona, Paola; Paglietti, Giuseppe; Luciani, R; Costi, M. P; Steania Ferrari, S. | |
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines | 1-gen-2014 | Loddo, R; Briguglio, Irene; Corona, Paola; Piras, Sandra; Loriga, M; Paglietti, G; Carta, Antonio; Sanna, G; Giliberti, G; Ibba, C; Farci, P; La Colla, P. | |
Benzotriazole: an overview on its versatile biological behaviour | 1-gen-2015 | Briguglio, Irene; Piras, Sandra; Corona, Paola; Gavini, Elisabetta; Nieddu, M; Boatto, Gianpiero; Carta, Antonio | |
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives | 1-gen-2015 | Briguglio, Irene; Loddo, Roberta; Laurini, Erik; Fermeglia, Maurizio; Piras, Sandra; Corona, Paola; Giunchedi, Paolo; Gavini, Elisabetta; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; La Colla, Paolo; Pricl, Sabrina; Carta, Antonio | |
A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems | 1-gen-2016 | Carta, Antonio; Briguglio, Irene; Piras, Sandra; Corona, Paola; Ibba, R.; Laurini, E.; Fermeglia, M.; Pricl, S.; Desideri, N.; Atzori, E. M.; La Colla, P.; Collu, G.; Delogu, I.; Loddo, R. | |
Synthesis of 2-(Quinoxalin-2-ylamino-benzotriazolyl) Pentanedioic Derivatives as Potential Anti-Folate Agents | 1-gen-2016 | Briguglio, Irene; Piras, Sandra; Corona, Paola; Pirisi, Maria Antonietta; Burrai, L; Boatto, Gianpiero; Gavini, Elisabetta; Rassu, Giovanna | |
Triazolopyridinyl-acrylonitrile derivatives as antimicrotubule agents: synthesis, in vitro and in silico characterization of antiproliferative activity, inhibition of tubulin polymerization and binding thermodynamics | 1-gen-2017 | Briguglio, Irene; Laurini, Erik; Pirisi, Maria Antonietta; Piras, Sandra; Corona, Paola; Fermeglia, Maurizio; Pricl, Sabrina; Carta, Antonio | |
Antiviral activities of 5-chlorobenzotriazole derivatives | 1-gen-2018 | Ibba, Roberta; Corona, P; Carta, A; Giunchedi, P; Loddo, R; Sanna, Giuseppina; Delogu, Ilenia; Piras, S | |
Quinoxaline derivatives as new inhibitors of coxsackievirus B5 | 1-gen-2018 | Carta, Antonio; Giuseppina, Sanna; Briguglio, Irene; Madeddu, Silvia; Vitale, Gabriella; Piras, Sandra; Corona, Paola; Peana, Alessandra Tiziana; Laurini, Erik; Fermeglia, Maurizio; Pricl, Sabrina; Alessandra, Serra; Carta, Elisa; Loddo, Roberta; Giliberti, Gabriele | |
Enhancement of antimicrobial activity of pump inhibitors associating drugs | 1-gen-2019 | Usai, Donatella; Donadu, Matthew; Bua, Alessandra; Molicotti, Paola; Zanetti, Stefania; Piras, Sandra; Corona, Paola; Ibba, Roberta; Carta, Antonio | |
Design, synthesis and antitubercular activity of 4-alkoxy-triazoloquinolones able to inhibit the M. tuberculosis DNA gyrase | 1-gen-2019 | Carta, Antonio; Bua, Alessandra; Corona, Paola; Piras, Sandra; Briguglio, Irene; Molicotti, Paola; Zanetti, Stefania; Laurini, Erik; Aulic, Suzana; Fermeglia, Maurizio; Pricl, Sabrina | |
Poly (ethyl 2-cyanoacrylate) nanoparticles (PECA-NPs) as possible agents in tumor treatment | 1-gen-2019 | Obinu, Antonella; Rassu, Giovanna; Corona, Paola; Maestri, Marcello; Riva, Federica; Miele, Dalila; Giunchedi, Paolo; Gavini, Elisabetta | |
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands | 1-gen-2019 | Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A. | |
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors | 1-gen-2019 | Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A. | |
Dichloro-phenyl -benzotriazoles: a new selective class of human respiratory syncytial virus entry inhibitors | 1-gen-2019 | Piras, Sandra; Sanna, Giuseppina; Carta, Antonio; Corona, Paola; Ibba, Roberta; Loddo, Roberta; Madeddu, Silvia; Caria, Paola; Aulic, Suzana; Laurini, Erik; Fermeglia, Maurizio; Pricl, Sabrina |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile