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Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties
2020-01-01 Weidong, L.; Sanna, L.; Bordoni, V.; Tiansheng, Z.; Chengxun, L.; Murineddu, G.; Pinna, G. A.; Kelvin, D. J.; Bagella, L.
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism
2016-01-01 Fois, G. R.; Fattore, L.; Murineddu, Gabriele; Salis, A.; Pintore, Giorgio Antonio Mario; Asproni, Battistina; Pinna, Gerard Aime; Diana, Marco
Thienocinnolinone alkanoic acid derivatives as aldose reductase inhibitors
2006-01-01 Pau, Amedeo; Asproni, Battistina; Murineddu, Gabriele; Boatto, Gianpiero; Grella, Giuseppe Enrico; Rakowitz, D.; Costantino, L.; Pinna, Gerard Aime
TRICYCLIC 3-(2H)-PYRIDAZINONE DERIVATIVES - SYNTHESIS AND EVALUATION OF THEIR ANTISECRETORY AND ANTIULCER ACTIVITY
1992-01-01 Cignarella, G.; Barlocco, D.; Villa, S.; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A.; Bestetti, A.
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction
2021-01-01 Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A.
Tricyclic pyrazoles Part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands
2014-01-01 Pinna, G; Curzu, Maria Michela; Dore, A; Lazzari, P; Ruiu, S; Pau, Amedeo; Murineddu, Gabriele; Pinna, Gerard Aime
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2 ',4 '-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyra zole-3-carboxamide
2006-01-01 Murineddu, Gabriele; Lazzari, P; Ruiu, S; Sanna, A; Loriga, G; Manca, I; Falzoi, M; Dessi, C; Curzu, Maria Michela; Chelucci, Giorgio Adolfo; Pani, L.; Pinna, Gerard Aime
Tricyclic pyrazoles. An Efficient approach to cannabinoid analogues with a tricyclic framework incorporating the pyrrole and pyrazole moieties
2012-01-01 Pinna, Gerard Aime; Chelucci, Giorgio Adolfo; Baldino, S.; Pinna, Giansalvo
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors
2003-01-01 Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzolglindazole-based ligands for cannabinoid receptors
2005-01-01 Murineddu, Gabriele; Rulu, S.; Mussinu, J. M.; Loriga, G.; Grella, G. E.; Caral, M. A. M.; Lazzarl, P.; Pani, L.; Pinna, Gerard Aime
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties | 1-gen-2020 | Weidong, L.; Sanna, L.; Bordoni, V.; Tiansheng, Z.; Chengxun, L.; Murineddu, G.; Pinna, G. A.; Kelvin, D. J.; Bagella, L. | |
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism | 1-gen-2016 | Fois, G. R.; Fattore, L.; Murineddu, Gabriele; Salis, A.; Pintore, Giorgio Antonio Mario; Asproni, Battistina; Pinna, Gerard Aime; Diana, Marco | |
Thienocinnolinone alkanoic acid derivatives as aldose reductase inhibitors | 1-gen-2006 | Pau, Amedeo; Asproni, Battistina; Murineddu, Gabriele; Boatto, Gianpiero; Grella, Giuseppe Enrico; Rakowitz, D.; Costantino, L.; Pinna, Gerard Aime | |
TRICYCLIC 3-(2H)-PYRIDAZINONE DERIVATIVES - SYNTHESIS AND EVALUATION OF THEIR ANTISECRETORY AND ANTIULCER ACTIVITY | 1-gen-1992 | Cignarella, G.; Barlocco, D.; Villa, S.; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A.; Bestetti, A. | |
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction | 1-gen-2021 | Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A. | |
Tricyclic pyrazoles Part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands | 1-gen-2014 | Pinna, G; Curzu, Maria Michela; Dore, A; Lazzari, P; Ruiu, S; Pau, Amedeo; Murineddu, Gabriele; Pinna, Gerard Aime | |
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2 ',4 '-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyra zole-3-carboxamide | 1-gen-2006 | Murineddu, Gabriele; Lazzari, P; Ruiu, S; Sanna, A; Loriga, G; Manca, I; Falzoi, M; Dessi, C; Curzu, Maria Michela; Chelucci, Giorgio Adolfo; Pani, L.; Pinna, Gerard Aime | |
Tricyclic pyrazoles. An Efficient approach to cannabinoid analogues with a tricyclic framework incorporating the pyrrole and pyrazole moieties | 1-gen-2012 | Pinna, Gerard Aime; Chelucci, Giorgio Adolfo; Baldino, S.; Pinna, Giansalvo | |
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors | 1-gen-2003 | Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime | |
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzolglindazole-based ligands for cannabinoid receptors | 1-gen-2005 | Murineddu, Gabriele; Rulu, S.; Mussinu, J. M.; Loriga, G.; Grella, G. E.; Caral, M. A. M.; Lazzarl, P.; Pani, L.; Pinna, Gerard Aime |
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Opzioni
Scopri
Tipologia
- 1 Contributo su Rivista 170
- 1 Contributo su Rivista::1.1 Arti... 170
Data di pubblicazione
- 2020 - 2023 6
- 2010 - 2019 50
- 2000 - 2009 52
- 1990 - 1999 44
- 1980 - 1989 16
- 1978 - 1979 2
Editore
- Pergamon / Elsevier 1
- Società chimica italiana 1
Rivista
- IL FARMACO 24
- EUROPEAN JOURNAL OF MEDICINAL CHE... 18
- TETRAHEDRON-ASYMMETRY 13
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- IL FARMACO. EDIZIONE SCIENTIFICA 7
- JOURNAL OF MEDICINAL CHEMISTRY 7
- MOLECULES 7
- TETRAHEDRON LETTERS 6
- JOURNAL OF HETEROCYCLIC CHEMISTRY 5
- SYNTHESIS 5
Keyword
- Drug Discovery3003 Pharmaceutical... 7
- Organic Chemistry 6
- Pharmacology 6
- Structure-Activity Relationship 6
- Cannabinoid 4
- Humans 4
- Molecular Medicine 4
- Receptor 4
- Synthesis 4
- 3 3
Lingua
- eng 108
- ita 2
Accesso al fulltext
- no fulltext 164
- open 6