RicercaInizia una nuova ricerca
NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
SYNTHESIS OF SOME 1-(3-HYDROXY-4-METHOXYBENZYL)-2-ALKYL-6,7-METHYLENEDIOXY-1,2,3,4-TETRAHY DROISOQUINOLINES AND THEIR BINDING AFFINITIES TO DA RECEPTOR SUBTYPES
1994-01-01 Pinna, Gerard Aime; Cignarella, G.; Scolastico, S.; Porceddu, M. L.
Synthesis of tricyclic condensed rings incorporating the pyrazole or isoxazole moieties bonded to a 4-piperidinyl substituent
2013-01-01 Pinna, G.; Loriga, G.; Pinna, G. A.; Chelucci, G.
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes
2020-01-01 Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A.
Synthesis, Modelling, and Antimitotic Properties of Tricyclic Systems Characterised by a 2-(5-Phenyl-1H-pyrrol-3-yl)-1,3,4-oxadiazole Moiety
2009-01-01 Pinna, Gerard Aime; Murineddu, Gabriele; Murruzzu, C.; Zuco, V.; Zunino, F.; Cappelletti, G.; Artali, R.; Cignarella, G.; Solano, L.; Villa, S.
Synthesis, modelling, and m-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes
2000-01-01 Pinna, Gerard Aime; Murineddu, Gabriele; M. M., Curzu; S., Villa; P., Vianello; P. A., Borea; S., Gessi; L., Toma; D., Colombo; G., Cignarella
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonists
2016-01-01 Dore, A.; Asproni, Battistina; Scampuddu, A.; Gessi, S.; Murineddu, Gabriele; Cichero, E.; Fossa, P.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime
Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes
2000-01-01 Vianello, P.; Albinati, A.; Pinna, Gerard Aime; Lavecchia, A.; Marinelli, L.; Borea, P. A.; Gessi, S.; Fadda, P.; Tronci, S.; Cignarella, G.
Synthesis, Pharmacological Evaluation and Docking Studies of Pyrrole Structure-Based CB2 Receptor Antagonists
2015-01-01 Ragusa, G; Gómez Cañas, M; Morales, P; Hurst, P. D. P.; Deligia, ; Pazos, F. R.; Pinna, Gerard Aime; Fernández Ruiz, J; Goya, P; Reggio, P. H.; Jagerovic, N; García Arencibia, M; Murineddu, Gabriele
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands
2018-01-01 Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele
Synthetic Methods for the Hydrodehalogenation of Halogenated Hetrerocycles
2012-01-01 Chelucci, Giorgio Adolfo; Baldinu, S; Pinna, Gerard Aime; Pinna, Giansalvo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
SYNTHESIS OF SOME 1-(3-HYDROXY-4-METHOXYBENZYL)-2-ALKYL-6,7-METHYLENEDIOXY-1,2,3,4-TETRAHY DROISOQUINOLINES AND THEIR BINDING AFFINITIES TO DA RECEPTOR SUBTYPES | 1-gen-1994 | Pinna, Gerard Aime; Cignarella, G.; Scolastico, S.; Porceddu, M. L. | |
Synthesis of tricyclic condensed rings incorporating the pyrazole or isoxazole moieties bonded to a 4-piperidinyl substituent | 1-gen-2013 | Pinna, G.; Loriga, G.; Pinna, G. A.; Chelucci, G. | |
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes | 1-gen-2020 | Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A. | |
Synthesis, Modelling, and Antimitotic Properties of Tricyclic Systems Characterised by a 2-(5-Phenyl-1H-pyrrol-3-yl)-1,3,4-oxadiazole Moiety | 1-gen-2009 | Pinna, Gerard Aime; Murineddu, Gabriele; Murruzzu, C.; Zuco, V.; Zunino, F.; Cappelletti, G.; Artali, R.; Cignarella, G.; Solano, L.; Villa, S. | |
Synthesis, modelling, and m-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes | 1-gen-2000 | Pinna, Gerard Aime; Murineddu, Gabriele; M. M., Curzu; S., Villa; P., Vianello; P. A., Borea; S., Gessi; L., Toma; D., Colombo; G., Cignarella | |
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonists | 1-gen-2016 | Dore, A.; Asproni, Battistina; Scampuddu, A.; Gessi, S.; Murineddu, Gabriele; Cichero, E.; Fossa, P.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime | |
Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes | 1-gen-2000 | Vianello, P.; Albinati, A.; Pinna, Gerard Aime; Lavecchia, A.; Marinelli, L.; Borea, P. A.; Gessi, S.; Fadda, P.; Tronci, S.; Cignarella, G. | |
Synthesis, Pharmacological Evaluation and Docking Studies of Pyrrole Structure-Based CB2 Receptor Antagonists | 1-gen-2015 | Ragusa, G; Gómez Cañas, M; Morales, P; Hurst, P. D. P.; Deligia, ; Pazos, F. R.; Pinna, Gerard Aime; Fernández Ruiz, J; Goya, P; Reggio, P. H.; Jagerovic, N; García Arencibia, M; Murineddu, Gabriele | |
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands | 1-gen-2018 | Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele | |
Synthetic Methods for the Hydrodehalogenation of Halogenated Hetrerocycles | 1-gen-2012 | Chelucci, Giorgio Adolfo; Baldinu, S; Pinna, Gerard Aime; Pinna, Giansalvo |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile
Opzioni
Scopri
Tipologia
- 1 Contributo su Rivista 170
- 1 Contributo su Rivista::1.1 Arti... 170
Data di pubblicazione
- 2020 - 2023 6
- 2010 - 2019 50
- 2000 - 2009 52
- 1990 - 1999 44
- 1980 - 1989 16
- 1978 - 1979 2
Editore
- Pergamon / Elsevier 1
- Società chimica italiana 1
Rivista
- IL FARMACO 24
- EUROPEAN JOURNAL OF MEDICINAL CHE... 18
- TETRAHEDRON-ASYMMETRY 13
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- IL FARMACO. EDIZIONE SCIENTIFICA 7
- JOURNAL OF MEDICINAL CHEMISTRY 7
- MOLECULES 7
- TETRAHEDRON LETTERS 6
- JOURNAL OF HETEROCYCLIC CHEMISTRY 5
- SYNTHESIS 5
Keyword
- Drug Discovery3003 Pharmaceutical... 7
- Organic Chemistry 6
- Pharmacology 6
- Structure-Activity Relationship 6
- Cannabinoid 4
- Humans 4
- Molecular Medicine 4
- Receptor 4
- Synthesis 4
- 3 3
Lingua
- eng 108
- ita 2
Accesso al fulltext
- no fulltext 164
- open 6