Sfoglia per Titolo
Tricyclic 3(2H)pyridazinone derivatives. Synthesis and pharmacological evaluation of their antiulcer and antisecretory activity
1992-01-01 Cignarella, G; Barlocco, D; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A; Bestetti, A.
TRICYCLIC 3-(2H)-PYRIDAZINONE DERIVATIVES - SYNTHESIS AND EVALUATION OF THEIR ANTISECRETORY AND ANTIULCER ACTIVITY
1992-01-01 Cignarella, G.; Barlocco, D.; Villa, S.; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A.; Bestetti, A.
Tricyclic condensed pyrazole derivatives as CB1inhibitors
2010-01-01 Lazzari, P.; Loriga, G.; Manca, I.; Pinna, Gerard Aime
Tricyclic pyrazole derivatives and microemulsions thereof as CB1 and/or CB2 inhibitors.
2010-01-01 Lazzari, P.; Loriga, G.; Manca, I.; Pinna, Gerard Aime
Tricyclic pyrazole derivatives as cannabinoid receptor antagonist
2005-01-01 Lazzari, P.; Ruiu, S.; Pinna, Gerard Aime; Murineddu, Gabriele
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction
2021-01-01 Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A.
Tricyclic pyrazoles Part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands
2014-01-01 Pinna, G; Curzu, Maria Michela; Dore, A; Lazzari, P; Ruiu, S; Pau, Amedeo; Murineddu, Gabriele; Pinna, Gerard Aime
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2 ',4 '-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyra zole-3-carboxamide
2006-01-01 Murineddu, Gabriele; Lazzari, P; Ruiu, S; Sanna, A; Loriga, G; Manca, I; Falzoi, M; Dessi, C; Curzu, Maria Michela; Chelucci, Giorgio Adolfo; Pani, L.; Pinna, Gerard Aime
Tricyclic pyrazoles. An Efficient approach to cannabinoid analogues with a tricyclic framework incorporating the pyrrole and pyrazole moieties
2012-01-01 Pinna, Gerard Aime; Chelucci, Giorgio Adolfo; Baldino, S.; Pinna, Giansalvo
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors
2003-01-01 Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzolglindazole-based ligands for cannabinoid receptors
2005-01-01 Murineddu, Gabriele; Rulu, S.; Mussinu, J. M.; Loriga, G.; Grella, G. E.; Caral, M. A. M.; Lazzarl, P.; Pani, L.; Pinna, Gerard Aime
Tricyclic pyrazoles. Part 3. Synthesis, biological evaluation and molecular modelling of analogues of the cannabinoid antagonist NESS 0327
2005-01-01 Murineddu, Gabriele; Ruiu, S; Loriga, G; Manca, I; Lazzari, P; Reali, R; Pani, L; Toma, L; Pinna, Ga
Tricyclic pyrazoles. Part 5. novel 1,4-Dihydroindeno[1,2-c]pyrazole CB2 ligands using molecular hybridization based on scaffold hopping
2012-01-01 Murineddu, Gabriele; Asproni, Battistina; Ruiu, S; Deligia, F; Falzoi, M; Pau, Amedeo; Thomas, Bf; Zhang, Y; Pinna, Gerard Aime; Pani, L; Lazzari, P.
Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazoles: A versatile architecture for CB2 selective ligands
2014-01-01 Pinna, Giovanni; Loriga, Giovanni; Lazzari, Paolo; Ruiu, Stefania; Falzoi, Matteo; Frau, Simona; Pau, Amedeo; Murineddu, Gabriele; Asproni, Battistina; Pinna, Gerard A.
Tricyclic Pyrazoles. Part 8. Synthesis, Biological Evaluation and Modelling of Tricyclic Pyrazole Carboxamides as Potential CB2 Receptor Ligands with Antagonist/Inverse Agonist Properties.
2016-01-01 Deiana, V; Gómez Cañas, M; Pazos, M. R.; Fernández Ruiz, J; Asproni, B; Cichero, E; Fossa, P; Muñoz, E; Deligia, F; Murineddu, Gabriele; García Arencibia, M; Pinna, Gerard Aime
Tricyclic pyrazoles: synthesis and biological evaluation of novel 4,5-dihydrobenzo-1h-6-oxa-cyclohepta[1,2-c] pyrazole-based analogues of the cannabinoid antagonist ness 0327
2008-01-01 Pau, Amedeo; Pinna, Gérard Aimé; Dessì, Cristian; Murruzzu, Caterina; Ruiu, Stefania; Lazzari, Paolo; Chelucci, Giorgio Adolfo; Reali, Roberta; Pani, Luca; Murineddu, Gabriele
Tricyclic pyridazines: a versatile substrate for cardiovascular compounds
1995-01-01 Cignarella, G; Curzu, M. M.; Pinna, Gerard Aime; Barlocco, D.
Tricyclic pyridazines: a versatile substrate for pharmacologically active compounds
1994-01-01 Cignarella, G.; Barlocco, D.; Pinna, Gerard Aime; Curzu, M. M.
Tricyclic structures related to antihypertensive and antithrombotic indenopyridazinones
1988-01-01 Cignarella, G; Barlocco, D; Pinna, Gerard Aime; Loriga, M; Curzu, M. M.; Tofanetti, O; Lumachi, B.
Tricyclic thieno-pyrazoles as new potent and selective CB2 ligands
2014-01-01 Dore, A; Pinna, G; Curzu, M. M.; Lazzari, P; Ruiu, S; Pau, A; Murineddu, Gabriele; Pinna, Gerard Aime
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Tricyclic 3(2H)pyridazinone derivatives. Synthesis and pharmacological evaluation of their antiulcer and antisecretory activity | 1-gen-1992 | Cignarella, G; Barlocco, D; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A; Bestetti, A. | |
TRICYCLIC 3-(2H)-PYRIDAZINONE DERIVATIVES - SYNTHESIS AND EVALUATION OF THEIR ANTISECRETORY AND ANTIULCER ACTIVITY | 1-gen-1992 | Cignarella, G.; Barlocco, D.; Villa, S.; Curzu, M. M.; Pinna, Gerard Aime; Lavezzo, A.; Bestetti, A. | |
Tricyclic condensed pyrazole derivatives as CB1inhibitors | 1-gen-2010 | Lazzari, P.; Loriga, G.; Manca, I.; Pinna, Gerard Aime | |
Tricyclic pyrazole derivatives and microemulsions thereof as CB1 and/or CB2 inhibitors. | 1-gen-2010 | Lazzari, P.; Loriga, G.; Manca, I.; Pinna, Gerard Aime | |
Tricyclic pyrazole derivatives as cannabinoid receptor antagonist | 1-gen-2005 | Lazzari, P.; Ruiu, S.; Pinna, Gerard Aime; Murineddu, Gabriele | |
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction | 1-gen-2021 | Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A. | |
Tricyclic pyrazoles Part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands | 1-gen-2014 | Pinna, G; Curzu, Maria Michela; Dore, A; Lazzari, P; Ruiu, S; Pau, Amedeo; Murineddu, Gabriele; Pinna, Gerard Aime | |
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2 ',4 '-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyra zole-3-carboxamide | 1-gen-2006 | Murineddu, Gabriele; Lazzari, P; Ruiu, S; Sanna, A; Loriga, G; Manca, I; Falzoi, M; Dessi, C; Curzu, Maria Michela; Chelucci, Giorgio Adolfo; Pani, L.; Pinna, Gerard Aime | |
Tricyclic pyrazoles. An Efficient approach to cannabinoid analogues with a tricyclic framework incorporating the pyrrole and pyrazole moieties | 1-gen-2012 | Pinna, Gerard Aime; Chelucci, Giorgio Adolfo; Baldino, S.; Pinna, Giansalvo | |
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors | 1-gen-2003 | Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime | |
Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzolglindazole-based ligands for cannabinoid receptors | 1-gen-2005 | Murineddu, Gabriele; Rulu, S.; Mussinu, J. M.; Loriga, G.; Grella, G. E.; Caral, M. A. M.; Lazzarl, P.; Pani, L.; Pinna, Gerard Aime | |
Tricyclic pyrazoles. Part 3. Synthesis, biological evaluation and molecular modelling of analogues of the cannabinoid antagonist NESS 0327 | 1-gen-2005 | Murineddu, Gabriele; Ruiu, S; Loriga, G; Manca, I; Lazzari, P; Reali, R; Pani, L; Toma, L; Pinna, Ga | |
Tricyclic pyrazoles. Part 5. novel 1,4-Dihydroindeno[1,2-c]pyrazole CB2 ligands using molecular hybridization based on scaffold hopping | 1-gen-2012 | Murineddu, Gabriele; Asproni, Battistina; Ruiu, S; Deligia, F; Falzoi, M; Pau, Amedeo; Thomas, Bf; Zhang, Y; Pinna, Gerard Aime; Pani, L; Lazzari, P. | |
Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazoles: A versatile architecture for CB2 selective ligands | 1-gen-2014 | Pinna, Giovanni; Loriga, Giovanni; Lazzari, Paolo; Ruiu, Stefania; Falzoi, Matteo; Frau, Simona; Pau, Amedeo; Murineddu, Gabriele; Asproni, Battistina; Pinna, Gerard A. | |
Tricyclic Pyrazoles. Part 8. Synthesis, Biological Evaluation and Modelling of Tricyclic Pyrazole Carboxamides as Potential CB2 Receptor Ligands with Antagonist/Inverse Agonist Properties. | 1-gen-2016 | Deiana, V; Gómez Cañas, M; Pazos, M. R.; Fernández Ruiz, J; Asproni, B; Cichero, E; Fossa, P; Muñoz, E; Deligia, F; Murineddu, Gabriele; García Arencibia, M; Pinna, Gerard Aime | |
Tricyclic pyrazoles: synthesis and biological evaluation of novel 4,5-dihydrobenzo-1h-6-oxa-cyclohepta[1,2-c] pyrazole-based analogues of the cannabinoid antagonist ness 0327 | 1-gen-2008 | Pau, Amedeo; Pinna, Gérard Aimé; Dessì, Cristian; Murruzzu, Caterina; Ruiu, Stefania; Lazzari, Paolo; Chelucci, Giorgio Adolfo; Reali, Roberta; Pani, Luca; Murineddu, Gabriele | |
Tricyclic pyridazines: a versatile substrate for cardiovascular compounds | 1-gen-1995 | Cignarella, G; Curzu, M. M.; Pinna, Gerard Aime; Barlocco, D. | |
Tricyclic pyridazines: a versatile substrate for pharmacologically active compounds | 1-gen-1994 | Cignarella, G.; Barlocco, D.; Pinna, Gerard Aime; Curzu, M. M. | |
Tricyclic structures related to antihypertensive and antithrombotic indenopyridazinones | 1-gen-1988 | Cignarella, G; Barlocco, D; Pinna, Gerard Aime; Loriga, M; Curzu, M. M.; Tofanetti, O; Lumachi, B. | |
Tricyclic thieno-pyrazoles as new potent and selective CB2 ligands | 1-gen-2014 | Dore, A; Pinna, G; Curzu, M. M.; Lazzari, P; Ruiu, S; Pau, A; Murineddu, Gabriele; Pinna, Gerard Aime |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile