Sfoglia per Autore
Synthesis of (2R,5S)- and (2S, SS)-2-Carboxy-l,4-diaza- [4.3.0]bicyclononane as Building Blocks for the Synthesis of New Potential HIV Protease Inhibitors.
1996-01-01 Porcheddu, Andrea; Giacomelli, G; Falorni, M.
General approach to the synthesis of optically active 2-carboxy-4-[3'- (diethoxyphosphinyl)propyl]-5-alkylpiperazines (CPP analogues)
1997-01-01 Porcheddu, Andrea; Falorni, M; Giacomelli, G.
New 1,3,5-triazine derivatives as templates for the homogeneous phase synthesis of chemical libraries
1998-01-01 Porcheddu, Andrea; Falorni, M; Giacomelli, Giampaolo; Mameli, L.
A Simple Method for the Reduction of Carboxylic Acids to Aldehydes or Alcohols Using H2 and Pd/C
1999-01-01 Porcheddu, Andrea; Taddei, M; Falorni, M; Giacomelli, G.
Preparazione di un nuovo reattivo supportato su fase solida per la realizzazione di reazioni radicaliche
2000-01-01 Porcheddu, Andrea; Porcu, Giancarlo; Giacomelli, Giampaolo; Taddei, Maurizio
DMTMM, un nuovo reattivo di "coupling" per la sintesi di ammidi in fase solida ed in fase omogenea
2000-01-01 Giacomelli, Giampaolo; Porcheddu, Andrea; Falchi, Alessandro; Taddei, Maurizio
4-(4,6-Dimethoxy[1,3,5]triazin-2-yl)-4-methyl morpholinium chloride (DMTMM): a valuable alternative to PyBOP for solid phase peptide synthesis
2000-01-01 Falchi, A.; Giacomelli, Giampaolo; Porcheddu, Andrea; Taddei, M.
Solution-Phase Syntesis of Mixed Amide Libraries by” Simultaneous Addition of Functionalities (SPSAF) to a Diketopiperazine Tetracarboxylic Acid Scaffold Monitored by GC Analysis of Isobutylic alcohol
2000-01-01 Falorni, M.; Giacomelli, G.; Porcheddu, Andrea; Taddei, M.
New Oxazole-Based Conformationally restricted Peptidomimetics: Design and Synthesis of a Pseudopeptide
2000-01-01 Dettori, G.; Falorni, M.; Giacomelli, G.; Porcheddu, Andrea
A valuable activating agent for carboxylic acids in solution, liquid and solid phase synthesis
2001-01-01 Porcheddu, Andrea; Taddei, M; Falchi, A.
Small Ring Constrained Peptidomimeics. Synthesis of Epoxy-Peptidomimetics Inhibitors of Cysteine Proteases
2001-01-01 Demarcus, M.; Ganadu, L. M.; Mura, G. M.; Porcheddu, Andrea; Quaranta, L.; Reginato, G.; Taddei, M.
A Mild and Efficient Alternative to the Classical Swern Oxidation
2001-01-01 DE LUCA, Lidia Vera Giovanna; Giacomelli, Giampaolo; Porcheddu, Andrea
Pirazoli ed isossazoli funzionalizzati: nuove strategie di sintesi
2002-01-01 De Luca, Lidia Vera Giovanna; Giacomelli, Giampaolo; Porcheddu, Andrea; Salaris, Margherita; Taddei, Maurizio
Triclorotriazina: un nuovo reattivo per antiche reazioni
2002-01-01 De Luca, Lidia Vera Giovanna; Giacomelli, Giampaolo; Porcheddu, Andrea
Cellulose Beads: a New Versatile Solid Support for Microwave- Assisted Synthesis. Preparation of Pyrazole and Isoxazole Libraries
2003-01-01 DE LUCA, Lidia Vera Giovanna; Giacomelli, Giampaolo; Porcheddu, Andrea; Salaris, M.; Taddei, M.
A NEW, RAPID, GENERAL PROCEDURE FOR THE SYNTHESIS OF ORGANIC MOLECULES SUPPORTED ON METHOXY-POLYETHYLENE GLYCOL (MEOPEG) UNDER MICROWAVE IRRADIATION CONDITIONS
2003-01-01 Porcheddu, Andrea; Ruda, G. F.; Sega, A.; Taddei, M.
Trichloroisocyanuric/TEMPO Oxidation of Alcohols under Mild Conditions: A Close Investigation
2003-01-01 DE LUCA, Lidia Vera Giovanna; Giacomelli, Giampaolo; Masala, M.; Porcheddu, Andrea
Simple One-Flask Method for the Preparation of Hydroxamic Acids
2003-01-01 Giacomelli, G.; Porcheddu, Andrea; Salaris, M.
Preparation of pyrazole and isoxazole libraries on cellulose beads: a new cheap and versatile biopolymer
2003-01-01 DE LUCA, Lidia Vera Giovanna; Giacomelli, G.; Porcheddu, Andrea; Salaris, M.; Taddei, M.
Microwave-Assisted Solution-Phase Synthesis of 1,4,5-Trisubstituted Pyrazoles
2003-01-01 Giacomelli, Giampaolo; Porcheddu, Andrea; Salaris, M.; Taddei, M.
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