Sfoglia per Autore
Single amino acid substitution in HIV-1 integrase catalytic core causes a dramatic shift in inhibitor selectivity
2008-01-01 Sechi, Mario; Al-Mawsawi, Laith Q.; Neamati, Nouri
Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors
2009-01-01 Sechi, Mario; Giuseppe, Rizzi; Alessia, Bacchi; Mauro, Carcelli; Dominga, Rogolino; Nicolino, Pala; TINO W., SANCHEZ C; Laleh, Taheri; Raveendra, Dayam; Nouri, Neamati
Synthesis and Evaluation of Different Fatty Acid Esters Formulated into Precirol (R) ATO-Based Lipid Nanoparticles as Vehicles for Topical Delivery
2009-01-01 Sanna, Vanna; Mariani, Alberto; Caria, Giuseppe; Sechi, Mario
Design, synthesis, molecular modeling and anti-HIV 1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes
2009-01-01 Sechi, Mario; Carta, Fabrizio; Sannia, Luciano; Dallocchio, Roberto; Dessi, Alessandro; Al Safi, Rasha I; Neamati, Nouri
Targeting HIV-1 Integrase Zinc Binding Motif. Chapter 37
2009-01-01 Sechi, Mario; Mauro, Carcelli; Dominga, Rogolino; Nouri, Neamati
DNA Binders: 1. Evaluation of DNA-Interactive Ability, Design, and Synthesis of Novel Intercalating Agents
2009-01-01 Sechi, Mario; Marco, Derudas; Roberto, Dallocchio; Alessandro, Dessì; Alessia, Cosseddu; Giuseppe, Paglietti
DNA Binders: 2. Molecular Recognition of DNA by 2,3,6,7-tetrahydro-1H-pyrrolo[1,2-a]indole-1,8(5H)-dione bis(4,5-dihydro-1H-imidazol-2-ylhydrazone) as a Prototype of “Two-Armed” Intercalating Agents
2009-01-01 Dallocchio, R; Dessì, A; Sanna, Vanna Annunziata; Pala, N; Campesi, Ilaria; Paglietti, G; Sechi, Mario
Investigation of furo[2,3-h]- and pyridazino[3,4-f]cinnolin-3-ol scaffolds as substrates for the development of novel HIV-1 integrase inhibitors
2011-01-01 Gomaa, M. F. Y.; Pala, Nicolino; Derudas, N; Hasanen, J. A. E.; El tamany, E. S. H.; Casule, P; Mariani, Alberto; Sechi, Mario
Design and Synthesis of Novel Polycycles Based on the 3H-pyrrolo/6,7-dihydropyrido[1,2-a]indole scaffold as Templates for Pharmaceutical Development
2011-01-01 Derudas, M; Pala, Nicolino; Sanna, Vanna Annunziata; Dallocchio, R; Dessì, A; Roggio, A. M.; Sechi, Mario
Oxidative stress and mitochondria damage contribute to silica nanoparticle-induced cytotoxicity in human endothelial cells
2011-01-01 Punzoni, S.; Sanna, Vanna Annunziata; Cossu, A.; Posadino, A. M.; Bandiera, Pasquale; Montella, Andrea Costantino Mario; Uzzau, Sergio; Sechi, Mario; Pintus, Gianfranco
Investigating the Role of Metal Chelation in HIV-1 Integrase Strand Transfer Inhibitors
2011-01-01 Bacchi, Alessia; Carcelli, Mauro; Compari, Carlotta; Fisicaro, Emilia; Pala, Nicolino; Rispoli, Gabriele; Rogolino, Dominga; Sanchez, Tino W; Sechi, Mario; Sinisi, Valentina; Neamati, Nouri
HIV-1 IN strand transfer inhibitors: a focus on metal binding
2011-01-01 Bacchi, Alessia; Carcelli, Mauro; Compari, Carlotta; Fisicaro, Emilia; Pala, Nicolino; Rispoli, Gabriele; Rogolino, Dominga; W. Sanchez, Tino; Sechi, Mario; Neamati, Nouri
Role of metals in HIV-1 integrase inhibitor design. Chapter 20
2011-01-01 Sechi, Mario; Mauro, Carcelli; Dominga, Rogolino; Nouri, Neamati
Valutazione in vitro della riflettività di nuovi prototipi di microbolle a rivestimento polimerico mediante l’impiego del software Qontrast
2011-01-01 Virgilio, G; Sanna, Vanna Annunziata; Scanu, D; Pintus, Gianfranco; Sirigu, D; Uzzau, Sergio; Marzo, M; Sechi, M; Migaleddu, V.
Sintesi di Idrogel di poli(N-Isopropilacrilammide) contenenti grafene ottenuti attraverso la tecnica della polimerizzazione frontal
2011-01-01 Alzari, Valeria; Nuvoli, Daniele; Sanna, R; Scognamillo, S; Piccinini, M; Gioffredi, E; Malucelli, G; Sechi, M; Sanna, V; Mariani, Alberto
Docetaxel-loaded nanoparticles based on PLA-co-caprolactone and PLGA-co-caprolactone for prostate cancer treatment
2011-01-01 Roggio, Am; Sanna, Vanna Annunziata; Posadino, Am; Cossu, A; Marceddu, S; Mariani, Alberto; Alzari, Valeria; Uzzau, Sergio; Pintus, Gf; Sechi, M.
Targeted Biocompatible Nanoparticles for tie Delivery of (-)-Epigallocatechin 3-Gallate to Prostate Cancer Cells
2011-01-01 Sanna, V; Pintus, Gianfranco; Roggio, Am; Punzoni, S; Posadino, Am; Arca, A; Marceddu, S; Bandiera, Pasquale; Uzzau, Sergio; Sechi, M.
Virtual Screening-Driven Identification of Human Carbonic Anhydrase Inhibitors incorporating an Original, New Pharmacophore
2011-01-01 Pala, Nicolino; Dallocchio, R; Dessi, A; Brancale, A; Carta, F; Ihm, S; Maresca, A; Sechi, Mario; Supuran, C. T.
Development of polymeric microbubbles targeted to prostate-specific membrane antigen as prototype of novel ultrasound contrast agents
2011-01-01 Sanna, Vanna Annunziata; Pintus, Gianfranco; Bandiera, Pasquale; Anedda, R.; Punzoni, S.; Sanna, B.; Migaleddu, V.; Uzzau, Sergio; Sechi, Mario
Novel docetaxel-loaded nanoparticles based on poly(lactide-co-caprolactone) and poly(lactideco-glycolide-co-caprolactone) for prostate cancer treatment: formulation, characterization, and cytotoxicity studies
2011-01-01 Sanna, Vanna Annunziata; Roggio, Am; Posadino, Am; Cossu, Annalisa; Marceddu, S; Mariani, Alberto; Alzari, Valeria; Uzzau, Sergio; Pintus, Gianfranco; Sechi, Mario
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Single amino acid substitution in HIV-1 integrase catalytic core causes a dramatic shift in inhibitor selectivity | 1-gen-2008 | Sechi, Mario; Al-Mawsawi, Laith Q.; Neamati, Nouri | |
Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors | 1-gen-2009 | Sechi, Mario; Giuseppe, Rizzi; Alessia, Bacchi; Mauro, Carcelli; Dominga, Rogolino; Nicolino, Pala; TINO W., SANCHEZ C; Laleh, Taheri; Raveendra, Dayam; Nouri, Neamati | |
Synthesis and Evaluation of Different Fatty Acid Esters Formulated into Precirol (R) ATO-Based Lipid Nanoparticles as Vehicles for Topical Delivery | 1-gen-2009 | Sanna, Vanna; Mariani, Alberto; Caria, Giuseppe; Sechi, Mario | |
Design, synthesis, molecular modeling and anti-HIV 1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes | 1-gen-2009 | Sechi, Mario; Carta, Fabrizio; Sannia, Luciano; Dallocchio, Roberto; Dessi, Alessandro; Al Safi, Rasha I; Neamati, Nouri | |
Targeting HIV-1 Integrase Zinc Binding Motif. Chapter 37 | 1-gen-2009 | Sechi, Mario; Mauro, Carcelli; Dominga, Rogolino; Nouri, Neamati | |
DNA Binders: 1. Evaluation of DNA-Interactive Ability, Design, and Synthesis of Novel Intercalating Agents | 1-gen-2009 | Sechi, Mario; Marco, Derudas; Roberto, Dallocchio; Alessandro, Dessì; Alessia, Cosseddu; Giuseppe, Paglietti | |
DNA Binders: 2. Molecular Recognition of DNA by 2,3,6,7-tetrahydro-1H-pyrrolo[1,2-a]indole-1,8(5H)-dione bis(4,5-dihydro-1H-imidazol-2-ylhydrazone) as a Prototype of “Two-Armed” Intercalating Agents | 1-gen-2009 | Dallocchio, R; Dessì, A; Sanna, Vanna Annunziata; Pala, N; Campesi, Ilaria; Paglietti, G; Sechi, Mario | |
Investigation of furo[2,3-h]- and pyridazino[3,4-f]cinnolin-3-ol scaffolds as substrates for the development of novel HIV-1 integrase inhibitors | 1-gen-2011 | Gomaa, M. F. Y.; Pala, Nicolino; Derudas, N; Hasanen, J. A. E.; El tamany, E. S. H.; Casule, P; Mariani, Alberto; Sechi, Mario | |
Design and Synthesis of Novel Polycycles Based on the 3H-pyrrolo/6,7-dihydropyrido[1,2-a]indole scaffold as Templates for Pharmaceutical Development | 1-gen-2011 | Derudas, M; Pala, Nicolino; Sanna, Vanna Annunziata; Dallocchio, R; Dessì, A; Roggio, A. M.; Sechi, Mario | |
Oxidative stress and mitochondria damage contribute to silica nanoparticle-induced cytotoxicity in human endothelial cells | 1-gen-2011 | Punzoni, S.; Sanna, Vanna Annunziata; Cossu, A.; Posadino, A. M.; Bandiera, Pasquale; Montella, Andrea Costantino Mario; Uzzau, Sergio; Sechi, Mario; Pintus, Gianfranco | |
Investigating the Role of Metal Chelation in HIV-1 Integrase Strand Transfer Inhibitors | 1-gen-2011 | Bacchi, Alessia; Carcelli, Mauro; Compari, Carlotta; Fisicaro, Emilia; Pala, Nicolino; Rispoli, Gabriele; Rogolino, Dominga; Sanchez, Tino W; Sechi, Mario; Sinisi, Valentina; Neamati, Nouri | |
HIV-1 IN strand transfer inhibitors: a focus on metal binding | 1-gen-2011 | Bacchi, Alessia; Carcelli, Mauro; Compari, Carlotta; Fisicaro, Emilia; Pala, Nicolino; Rispoli, Gabriele; Rogolino, Dominga; W. Sanchez, Tino; Sechi, Mario; Neamati, Nouri | |
Role of metals in HIV-1 integrase inhibitor design. Chapter 20 | 1-gen-2011 | Sechi, Mario; Mauro, Carcelli; Dominga, Rogolino; Nouri, Neamati | |
Valutazione in vitro della riflettività di nuovi prototipi di microbolle a rivestimento polimerico mediante l’impiego del software Qontrast | 1-gen-2011 | Virgilio, G; Sanna, Vanna Annunziata; Scanu, D; Pintus, Gianfranco; Sirigu, D; Uzzau, Sergio; Marzo, M; Sechi, M; Migaleddu, V. | |
Sintesi di Idrogel di poli(N-Isopropilacrilammide) contenenti grafene ottenuti attraverso la tecnica della polimerizzazione frontal | 1-gen-2011 | Alzari, Valeria; Nuvoli, Daniele; Sanna, R; Scognamillo, S; Piccinini, M; Gioffredi, E; Malucelli, G; Sechi, M; Sanna, V; Mariani, Alberto | |
Docetaxel-loaded nanoparticles based on PLA-co-caprolactone and PLGA-co-caprolactone for prostate cancer treatment | 1-gen-2011 | Roggio, Am; Sanna, Vanna Annunziata; Posadino, Am; Cossu, A; Marceddu, S; Mariani, Alberto; Alzari, Valeria; Uzzau, Sergio; Pintus, Gf; Sechi, M. | |
Targeted Biocompatible Nanoparticles for tie Delivery of (-)-Epigallocatechin 3-Gallate to Prostate Cancer Cells | 1-gen-2011 | Sanna, V; Pintus, Gianfranco; Roggio, Am; Punzoni, S; Posadino, Am; Arca, A; Marceddu, S; Bandiera, Pasquale; Uzzau, Sergio; Sechi, M. | |
Virtual Screening-Driven Identification of Human Carbonic Anhydrase Inhibitors incorporating an Original, New Pharmacophore | 1-gen-2011 | Pala, Nicolino; Dallocchio, R; Dessi, A; Brancale, A; Carta, F; Ihm, S; Maresca, A; Sechi, Mario; Supuran, C. T. | |
Development of polymeric microbubbles targeted to prostate-specific membrane antigen as prototype of novel ultrasound contrast agents | 1-gen-2011 | Sanna, Vanna Annunziata; Pintus, Gianfranco; Bandiera, Pasquale; Anedda, R.; Punzoni, S.; Sanna, B.; Migaleddu, V.; Uzzau, Sergio; Sechi, Mario | |
Novel docetaxel-loaded nanoparticles based on poly(lactide-co-caprolactone) and poly(lactideco-glycolide-co-caprolactone) for prostate cancer treatment: formulation, characterization, and cytotoxicity studies | 1-gen-2011 | Sanna, Vanna Annunziata; Roggio, Am; Posadino, Am; Cossu, Annalisa; Marceddu, S; Mariani, Alberto; Alzari, Valeria; Uzzau, Sergio; Pintus, Gianfranco; Sechi, Mario |
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