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An overview on different classes of viral entry and respiratory syncitial virus (RSV) fusion inhibitors
2010-01-01 Murineddu, Gabriele; Murruzzu, C.; Pinna, Gerard Aime
ANTIHYPERTENSIVE AND ANTITHROMBOTIC ACTIVITIES OF 6-(SUBSTITUTED PHENYL)-5-HYDROXYMETHYL-4,5-DIHYDRO-3(2H)PYRIDAZINONES
1987-01-01 Barlocco, D.; Martini, A.; Pinna, Gerard Aime; Curzu, M. M.; Sala, F.; Germini, M.
Application of an unusual ninhydrin-based reaction for the indirect chiral resolution of D,L-penicillamine
2011-01-01 Sotgia, S; Zinellu, Angelo; Pinna, Gerard Aime; Deiana, L.; Carru, Ciriaco
Behavior of 5,6-dihydrobenzo[h]cinnolinones towards hydrazine. Synthesis of benzo[h]cinnolinones and of 4-aminobenzo[h]cinnolinones
1999-01-01 Villa, S.; Evoli, G. L.; Cignarella, G.; Curzu, M. M.; Pinna, Gerard Aime
Behaviour of 5,6-dihydrothieno[2,3-h]cinnolin-3(2H)-one and 5,6-dihydrothieno[3,2-h]cinnolin-3(2H)-one towards hydrazine. Synthesis of thienocinnolinones and of 4-aminothienocinnolinones
1999-01-01 Villa, S.; Cignarella, G.; Curzu, M. M.; Pinna, Gerard Aime; Pini, E.; Toma, L.
Benzocondensed derivatives as rigid analogues of the mu-opioid agonist 3(8)-cinnamyl-8(3)-propionyl-3,8-diazabicyclo[3.2.1]octanes: synthesis, modeling, and affinity
1998-01-01 Cignarella, G.; Barlocco, D.; Vianello, P.; Villa, S.; Pinna, Gerard Aime; Fadda, P.; Fratta, W.; Toma, L.; Gessi, S.
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. .
2021-01-01 Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime
Chemistry of tricyclic-based heterocycles as useful scaffolds for phosphodiesterase 10A ligands
2013-01-01 Asproni, Battistina; Dore, A; Murineddu, Gabriele; Pinna, Gerard Aime
Chiral 2-(2-phenylthiophenyl)-5,6,7,8-tetrahydroquinolines: new N-S ligands for asymmetric catalysis - Palladium-catalyzed allylic alkylation and copper-catalyzed cyclopropanation reactions
2003-01-01 Chelucci, Giorgio Adolfo; Muroni, D.; Pinna, Gerard Aime; Saba, A.; Vignola, D.
Chiral 8-Amino Substituted 2-Phenyl-5,6,7,8-tetrahydro-6,6-dimethylmathanoquinolines as Chiral Ligands for Enantioselective Catalysis: Palladium Catalysed Allylic Substitution and Addition of Diethylzinc to Benzaldehyde
1997-01-01 Chelucci, Giorgio Adolfo; Pinna, Gerard Aime
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Tipologia
- 1 Contributo su Rivista 170
- 1 Contributo su Rivista::1.1 Arti... 170
Data di pubblicazione
- 2020 - 2023 6
- 2010 - 2019 50
- 2000 - 2009 52
- 1990 - 1999 44
- 1980 - 1989 16
- 1978 - 1979 2
Editore
- Pergamon / Elsevier 1
- Società chimica italiana 1
Rivista
- IL FARMACO 24
- EUROPEAN JOURNAL OF MEDICINAL CHE... 18
- TETRAHEDRON-ASYMMETRY 13
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- IL FARMACO. EDIZIONE SCIENTIFICA 7
- JOURNAL OF MEDICINAL CHEMISTRY 7
- MOLECULES 7
- TETRAHEDRON LETTERS 6
- JOURNAL OF HETEROCYCLIC CHEMISTRY 5
- SYNTHESIS 5
Keyword
- Drug Discovery3003 Pharmaceutical... 7
- Organic Chemistry 6
- Pharmacology 6
- Structure-Activity Relationship 6
- Cannabinoid 4
- Humans 4
- Molecular Medicine 4
- Receptor 4
- Synthesis 4
- 3 3
Lingua
- eng 108
- ita 2
Accesso al fulltext
- no fulltext 164
- open 6