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H2S-BASED THERAPEUTIC AGENTS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES 1-gen-2019 Calderone, Vincenzo; Puricelli, Guido; Rapposelli, Simona; Sestito, Simona
Epibatidine: A Promising Natural Alkaloid in Health 1-gen-2019 Salehi, Bahare; Sestito, Simona; Rapposelli, Simona; Peron, Gregorio; Calina, Daniela; Sharifi-Rad, Mehdi; Sharopov, Farukh; Martins, Natália; Sharifi-Rad, Javad
Memantine prodrug as a new agent for alzheimer’s disease 1-gen-2019 Sestito, S.; Daniele, S.; Pietrobono, D.; Citi, V.; Bellusci, L.; Chiellini, G.; Calderone, V.; Martini, C.; Rapposelli, S.
Multi-targeted ChEI-copper chelating molecules as neuroprotective agents 1-gen-2019 Sestito, Simona; Wang, Shengnan; Chen, Qiuhe; Lu, Junfeng; Bertini, Simone; Pomelli, Christian; Chiellini, Grazia; He, Xixin; Pi, Rongbiao; Rapposelli, Simona
A patent update on PDK1 inhibitors (2015-present) 1-gen-2019 Sestito, S.; Rapposelli, S.
Preclinical validation of 3-phosphoinositide-dependent protein kinase 1 inhibition in pancreatic cancer 1-gen-2019 Emmanouilidi, A.; Fyffe, C. A.; Ferro, R.; Edling, C. E.; Capone, E.; Sestito, S.; Rapposelli, S.; Lattanzio, R.; Iacobelli, S.; Sala, G.; Maffucci, T.; Falasca, M.
Design and synthesis of H2S-donor hybrids: A new treatment for Alzheimer's disease? 1-gen-2019 Sestito, S.; Pruccoli, L.; Runfola, M.; Citi, V.; Martelli, A.; Saccomanni, G.; Calderone, V.; Tarozzi, A.; Rapposelli, S.
Dual PDK1/aurora kinase a inhibitors reduce pancreatic cancer cell proliferation and colony formation 1-gen-2019 Casari, I.; Domenichini, A.; Sestito, S.; Capone, E.; Sala, G.; Rapposelli, S.; Falasca, M.
Collecting data through high throughput in vitro early toxicity and off-target liability assays to rapidly identify limitations of novel thyromimetics 1-gen-2020 Runfola, M.; Sestito, S.; Gul, S.; Chiellini, G.; Rapposelli, S.
3-Iodothyronamine and Derivatives: New Allies Against Metabolic Syndrome? 1-gen-2020 Rutigliano, Grazia; Bandini, Lavinia; Sestito, Simona; Chiellini, Grazia
Selective Thyroid Hormone Receptor-Beta (TRβ) Agonists: New Perspectives for the Treatment of Metabolic and Neurodegenerative Disorders 1-gen-2020 Saponaro, F.; Sestito, S.; Runfola, M.; Rapposelli, S.; Chiellini, G.
Turmeric and Its Major Compound Curcumin on Health: Bioactive Effects and Safety Profiles for Food, Pharmaceutical, Biotechnological and Medicinal Applications 1-gen-2020 Sharifi-Rad, J.; Rayess, Y. E.; Rizk, A. A.; Sadaka, C.; Zgheib, R.; Zam, W.; Sestito, S.; Rapposelli, S.; Neffe-Skocinska, K.; Zielinska, D.; Salehi, B.; Setzer, W. N.; Dosoky, N. S.; Taheri, Y.; El Beyrouthy, M.; Martorell, M.; Ostrander, E. A.; Suleria, H. A. R.; Cho, W. C.; Maroyi, A.; Martins, N.
Areca catechu—From farm to food and biomedical applications 1-gen-2020 Salehi, B.; Konovalov, D. A.; Fru, P.; Kapewangolo, P.; Peron, G.; Ksenija, M. S.; Cardoso, S. M.; Pereira, O. R.; Nigam, M.; Nicola, S.; Pignata, G.; Rapposelli, S.; Sestito, S.; Anil Kumar, N. V.; de la Luz Cadiz-Gurrea, M.; Segura-Carretero, A.; P. Mishra, A.; Sharifi-Rad, M.; C. Cho, W.; Taheri, Y.; Setzer, W. N.; Sharifi-Rad, J.
Design, synthesis and biological evaluation of novel TRβ selective agonists sustained by ADME-toxicity analysis 1-gen-2020 Runfola, Massimiliano; Sestito, Simona; Bellusci, Lorenza; La Pietra, Valeria; D'Amore, Vincenzo Maria; Kowalik, Marta Anna; Chiellini, Grazia; Gul, Sheraz; Perra, Andrea; Columbano, Amedeo; Marinelli, Luciana; Novellino, Ettore; Rapposelli, Simona
Endogenous 3-iodothyronamine (T1Am) and synthetic thyronamine-like analog SG-2 act as novel pleiotropic neuroprotective agents through the modulation of SIRT6 1-gen-2020 Bellusci, L.; Runfola, M.; Carnicelli, V.; Sestito, S.; Fulceri, F.; Santucci, F.; Lenzi, P.; Fornai, F.; Rapposelli, S.; Origlia, N.; Zucchi, R.; Chiellini, G.
ACE2 in the Era of SARS-CoV-2: Controversies and Novel Perspectives 1-gen-2020 Saponaro, F.; Rutigliano, G.; Sestito, S.; Bandini, L.; Storti, B.; Bizzarri, R.; Zucchi, R.
Potential role of two novel agonists of thyroid hormone receptor-β on liver regeneration 1-gen-2020 Perra, A.; Kowalik, M. A.; Cabras, L.; Runfola, M.; Sestito, S.; Migliore, C.; Giordano, S.; Chiellini, G.; Rapposelli, S.; Columbano, A.
A comprehensive assessment of a new series of 5′,6′-difluorobenzotriazole-acrylonitrile derivatives as microtubule targeting agents (MTAs) 1-gen-2021 Riu, F.; Sanna, L.; Ibba, R.; Piras, S.; Bordoni, V.; Scorciapino, M. A.; Lai, M.; Sestito, S.; Bagella, L.; Carta, A.
Inhibition of Enterovirus A71 by a Novel 2-Phenyl-Benzimidazole Derivative 1-gen-2021 Ibba, R.; Carta, A.; Madeddu, S.; Caria, P.; Serreli, G.; Piras, S.; Sestito, S.; Loddo, R.; Sanna, G.
Chitosan nanoparticles as a promising tool in nanomedicine with particular emphasis on oncological treatment 1-gen-2021 Sharifi-Rad, Javad; Quispe, Cristina; Butnariu, Monica; Rotariu, Lia Sanda; Sytar, Oksana; Sestito, Simona; Rapposelli, Simona; Akram, Muhammad; Iqbal, Mehwish; Krishna, Akash; Kumar, Nanjangud Venkatesh Anil; Braga, Susana S; Cardoso, Susana M; Jafernik, Karolina; Ekiert, Halina; Cruz-Martins, Natália; Szopa, Agnieszka; Villagran, Marcelo; Mardones, Lorena; Martorell, Miquel; Docea, Anca Oana; Calina, Daniela
Mostrati risultati da 21 a 40 di 47
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