Sfoglia per Autore
N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as μ-opioid receptor agonists. Effects on μ-affinity of arylalkenyl chain modifications
2002-01-01 Pinna, Gerard Aime; Cignarella, G.; Loriga, G.; Murineddu, Gabriele; Mussinu, J. M.; Ruiu, S.; Fadda, P.; Fratta, W.
Synthesis and D2-like binding affinity of new derivatives of N-(1-ethyl-2-pyrrolidinylmethyl)-4,5-dihydro-1H-benzo[g]indole-3-carboxamide and related 4H-[1]Benzothiopyrano[4,3-b]pyrrole and 5,6-Dihydro-4H benzo[6,7]cyclohepta[b]pyrrole-3-carboxamide Analogues
2002-01-01 Pinna, Gerard Aime; Pirisi, Ma; Chelucci, Giorgio Adolfo; Mussinu, Jm; Murineddu, Gabriele; Loriga, G; D'Aquila, Paolo Stefano; Serra, G.
Synthesis and cytotoxicity evaluation of thiophene analogues of 1-methyl-2,3-bis(hydroxymethyl)benzo[g]indole bis[N-(2-propyl)carbamate]
2002-01-01 Pirisi, Maria Antonietta; Murineddu, Gabriele; Mussinu, J. M.; Pinna, Gerard Aime
Oxadiazoles having antiproliferative activity
2003-01-01 Cignarella, G.; Pinna, G.; Murineddu, Gabriele
Oxadiazoles having anti proliferative activity
2003-01-01 Cignarella, G; Pinna, Gerard Aime; Murineddu, Gabriele
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors
2003-01-01 Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime
Synthesis of novel diazatricyclodecanes (DTDs). Effects of structural variation at the C3 ' allyl end and at the phenyl ring of the cinnamyl chain on mu-receptor affinity and opioid antinociception
2003-01-01 Pinna, Gerard Aime; Cignarella, G.; Ruiu, S.; Loriga, G.; Murineddu, Gabriele; Villa, S.; Grella, G. E.; Cossu, G.; Fratta, W.
Synthesis and cytotoxicity of substituted 2-benzylnaphth[2,3-d]imidazoles
2003-01-01 Grella, G. E.; Cabras, M. C.; Murineddu, Gabriele; Pau, Amedeo; Pinna, Gerard Aime
Synthesis of chiral C2-symmetric 1,10-phenanthrolines from naturally occurring monoterpenes
2003-01-01 Chelucci, Giorgio Adolfo; Loriga, G.; Murineddu, Gabriele; Pinna, Gerard Aime
Chromophore-modified bis-benzo[g]indazole carboxamides: synthesis and antiproliferactive activity of bis-benzo[g]indazole carboxamides and related dimers
2003-01-01 Pinna, Gerard Aime; Pirisi, Maria Antonietta; Mussinu, J. M.; Murineddu, Gabriele; Loriga, G.; Pau, Amedeo; Grella, G. E.
I 3,6-diazabiciclo[3.1.1]eptani: una nuova serie di potenti agonisti per i recettori µ degli oppioidi
2004-01-01 Pinna, Gérard Aimé; Loriga, Giovanni; Chelucci, Giorgio Adolfo; Murineddu, Gabriele; Ruiu, Stefania; Cignarella, Giorgio
I 3,6-diazabiciclo[3.1.1]eptani: una nuova serie di potenti agonisti per i recettori μ degli oppioidi
2004-01-01 Loriga, G; Ruiu, S; Murineddu, Gabriele; Chelucci, Giorgio Adolfo; Cignarella, G; Pinna, Gerard Aime
Composti farmaceutici
2004-01-01 Lazzari, P.; Ruiu, S.; Pinna, G. A.; Murineddu, Gabriele
Chiral pyridine N-oxides useful ligands for asymmetric catalysis
2004-01-01 Chelucci, Giorgio Adolfo; Murineddu, Gabriele; Pinna, Gerard Aime
Synthesis and cytotoxic activities of 3-(5-phenyl-[1.3.4]oxadiazol-2-yl)-1H-benzo[g]indole and related compounds
2005-01-01 Villa, S.; Solano, L.; Cignarella, G.; Murineddu, Gabriele; Pinna, Gerard Aime
Tricyclic pyrazole derivatives as cannabinoid receptor antagonist
2005-01-01 Lazzari, P.; Ruiu, S.; Pinna, Gerard Aime; Murineddu, Gabriele
Pharmaceutical compounds
2005-01-01 Murineddu, Gabriele; Ruiu, S; Lazzari, P; Pinna, Gerard Aime
Pharmaceutical compounds
2005-01-01 Lazzari, P; Ruiu, S; Pinna, Gerard Aime; Murineddu, Gabriele
Pyrazole derivatives having affinity for CB1 and/or CB2 receptors
2005-01-01 Lazzari, P; Ruiu, S; Pinna, Gerard Aime; Murineddu, Gabriele
Pharmaceutical compounds
2005-01-01 Lazzari, Paolo; Ruiu, Stefania; Pinna, ; Gerard, Aime; Murineddu, Gabriele; Gabriele,
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as μ-opioid receptor agonists. Effects on μ-affinity of arylalkenyl chain modifications | 1-gen-2002 | Pinna, Gerard Aime; Cignarella, G.; Loriga, G.; Murineddu, Gabriele; Mussinu, J. M.; Ruiu, S.; Fadda, P.; Fratta, W. | |
Synthesis and D2-like binding affinity of new derivatives of N-(1-ethyl-2-pyrrolidinylmethyl)-4,5-dihydro-1H-benzo[g]indole-3-carboxamide and related 4H-[1]Benzothiopyrano[4,3-b]pyrrole and 5,6-Dihydro-4H benzo[6,7]cyclohepta[b]pyrrole-3-carboxamide Analogues | 1-gen-2002 | Pinna, Gerard Aime; Pirisi, Ma; Chelucci, Giorgio Adolfo; Mussinu, Jm; Murineddu, Gabriele; Loriga, G; D'Aquila, Paolo Stefano; Serra, G. | |
Synthesis and cytotoxicity evaluation of thiophene analogues of 1-methyl-2,3-bis(hydroxymethyl)benzo[g]indole bis[N-(2-propyl)carbamate] | 1-gen-2002 | Pirisi, Maria Antonietta; Murineddu, Gabriele; Mussinu, J. M.; Pinna, Gerard Aime | |
Oxadiazoles having antiproliferative activity | 1-gen-2003 | Cignarella, G.; Pinna, G.; Murineddu, Gabriele | |
Oxadiazoles having anti proliferative activity | 1-gen-2003 | Cignarella, G; Pinna, Gerard Aime; Murineddu, Gabriele | |
Tricyclic pyrazoles. part 1: Synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1 and CB2 cannabinoid receptors | 1-gen-2003 | Mussinu, Jm; Ruiu, S; Mulè, Ac; Pau, A; Carai, Mam; Loriga, G; Murineddu, Gabriele; Pinna, Gerard Aime | |
Synthesis of novel diazatricyclodecanes (DTDs). Effects of structural variation at the C3 ' allyl end and at the phenyl ring of the cinnamyl chain on mu-receptor affinity and opioid antinociception | 1-gen-2003 | Pinna, Gerard Aime; Cignarella, G.; Ruiu, S.; Loriga, G.; Murineddu, Gabriele; Villa, S.; Grella, G. E.; Cossu, G.; Fratta, W. | |
Synthesis and cytotoxicity of substituted 2-benzylnaphth[2,3-d]imidazoles | 1-gen-2003 | Grella, G. E.; Cabras, M. C.; Murineddu, Gabriele; Pau, Amedeo; Pinna, Gerard Aime | |
Synthesis of chiral C2-symmetric 1,10-phenanthrolines from naturally occurring monoterpenes | 1-gen-2003 | Chelucci, Giorgio Adolfo; Loriga, G.; Murineddu, Gabriele; Pinna, Gerard Aime | |
Chromophore-modified bis-benzo[g]indazole carboxamides: synthesis and antiproliferactive activity of bis-benzo[g]indazole carboxamides and related dimers | 1-gen-2003 | Pinna, Gerard Aime; Pirisi, Maria Antonietta; Mussinu, J. M.; Murineddu, Gabriele; Loriga, G.; Pau, Amedeo; Grella, G. E. | |
I 3,6-diazabiciclo[3.1.1]eptani: una nuova serie di potenti agonisti per i recettori µ degli oppioidi | 1-gen-2004 | Pinna, Gérard Aimé; Loriga, Giovanni; Chelucci, Giorgio Adolfo; Murineddu, Gabriele; Ruiu, Stefania; Cignarella, Giorgio | |
I 3,6-diazabiciclo[3.1.1]eptani: una nuova serie di potenti agonisti per i recettori μ degli oppioidi | 1-gen-2004 | Loriga, G; Ruiu, S; Murineddu, Gabriele; Chelucci, Giorgio Adolfo; Cignarella, G; Pinna, Gerard Aime | |
Composti farmaceutici | 1-gen-2004 | Lazzari, P.; Ruiu, S.; Pinna, G. A.; Murineddu, Gabriele | |
Chiral pyridine N-oxides useful ligands for asymmetric catalysis | 1-gen-2004 | Chelucci, Giorgio Adolfo; Murineddu, Gabriele; Pinna, Gerard Aime | |
Synthesis and cytotoxic activities of 3-(5-phenyl-[1.3.4]oxadiazol-2-yl)-1H-benzo[g]indole and related compounds | 1-gen-2005 | Villa, S.; Solano, L.; Cignarella, G.; Murineddu, Gabriele; Pinna, Gerard Aime | |
Tricyclic pyrazole derivatives as cannabinoid receptor antagonist | 1-gen-2005 | Lazzari, P.; Ruiu, S.; Pinna, Gerard Aime; Murineddu, Gabriele | |
Pharmaceutical compounds | 1-gen-2005 | Murineddu, Gabriele; Ruiu, S; Lazzari, P; Pinna, Gerard Aime | |
Pharmaceutical compounds | 1-gen-2005 | Lazzari, P; Ruiu, S; Pinna, Gerard Aime; Murineddu, Gabriele | |
Pyrazole derivatives having affinity for CB1 and/or CB2 receptors | 1-gen-2005 | Lazzari, P; Ruiu, S; Pinna, Gerard Aime; Murineddu, Gabriele | |
Pharmaceutical compounds | 1-gen-2005 | Lazzari, Paolo; Ruiu, Stefania; Pinna, ; Gerard, Aime; Murineddu, Gabriele; Gabriele, |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile