Sfoglia per Autore
Design, Synthesis, and Antiviral Activities of New Benzotriazole-Based Derivatives
2023-01-01 Ibba, Roberta; Corona, Paola; Nonne, Francesca; Caria, Paola; Serreli, Gabriele; Palmas, Vanessa; Riu, Federico; Sestito, Simona; Nieddu, Maria; Loddo, Roberta; Sanna, Giuseppina; Piras, Sandra; Carta, Antonio
Improving in vivo oral bioavailability of a poorly soluble drug: a case study on polymeric versus lipid nanoparticles
2023-01-01 Rassu, Giovanna; Obinu, Antonella; Serri, Carla; Piras, Sandra; Carta, Antonio; Ferraro, Luca; Gavini, Elisabetta; Giunchedi, Paolo; Dalpiaz, Alessandro
Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication
2022-01-01 Ibba, Roberta; Riu, Federico; Delogu, Ilenia; Lupinu, Ilenia; Carboni, Gavino; Loddo, Roberta; Piras, Sandra; Carta, Antonio
A Lead-Based Fragment Library Screening of the Glycosyltransferase WaaG from Escherichia coli
2022-01-01 Riu, Federico; Ruda, Alessandro; Engström, Olof; Muheim, Claudio; Mobarak, Hani; Ståhle, Jonas; Kosma, Paul; Carta, Antonio; Daley, Daniel O; Widmalm, Göran
Quinoxaline-based efflux pump inhibitors restore drug susceptibility in drug-resistant nontuberculous mycobacteria
2022-01-01 Corona, Paola; Ibba, Roberta; Piras, Sandra; Molicotti, Paola; Bua, Alessandra; Carta, Antonio
Design, synthesis, and biological screening of a series of 4 '-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs)
2022-01-01 Riu, F; Ibba, R; Zoroddu, S; Sestito, S; Lai, M; Piras, S; Sanna, L; Bordoni, V; Bagella, L; Carta, A
Design, synthesis, and biological screening of a series of 4′-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs)
2022-01-01 Riu, Federico; Ibba, Roberta; Zoroddu, Stefano; Sestito, Simona; Lai, Michele; Piras, Sandra; Sanna, Luca; Bordoni, Valentina; Bagella, Luigi Marco; Carta, Antonio
Antibiotics and Carbohydrate-Containing Drugs Targeting Bacterial Cell Envelopes: An Overview
2022-01-01 Riu, Federico; Ruda, Alessandro; Ibba, Roberta; Sestito, Simona; Lupinu, Ilenia; Piras, Sandra; Widmalm, Göran; Carta, Antonio
Human Enterovirus B: Selective Inhibition by Quinoxaline Derivatives and Bioinformatic RNA-Motif Identification as New Targets
2022-01-01 Madeddu, Silvia; Ibba, Roberta; Sanna, Giuseppina; Piras, Sandra; Riu, Federico; Marongiu, Alessandra; Ambrosino, Annalisa; Caria, Paola; Onnis, Valentina; Franci, Gianluigi; Manzin, Aldo; Carta, Antonio
Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives
2021-01-01 Ibba, R.; Piras, S.; Corona, P.; Riu, F.; Loddo, R.; Delogu, I.; Collu, G.; Sanna, G.; Caria, P.; Dettori, T.; Carta, A.
Inhibition of Enterovirus A71 by a Novel 2-Phenyl-Benzimidazole Derivative
2021-01-01 Ibba, R.; Carta, A.; Madeddu, S.; Caria, P.; Serreli, G.; Piras, S.; Sestito, S.; Loddo, R.; Sanna, G.
A comprehensive assessment of a new series of 5′,6′-difluorobenzotriazole-acrylonitrile derivatives as microtubule targeting agents (MTAs)
2021-01-01 Riu, F.; Sanna, L.; Ibba, R.; Piras, S.; Bordoni, V.; Scorciapino, M. A.; Lai, M.; Sestito, S.; Bagella, L.; Carta, A.
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. .
2021-01-01 Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime
anti-BVDV Activity evaluation of Naphthoimidazole derivatives compared with parentalimidazoquinoline compounds
2020-01-01 Ibba, Roberta; Piras, Sandra; Delogu, Ilenia; Loddo, Roberta; Carta, Antonio
Phytochemical compositions and biological activities of essential oils from the leaves, rhizomes and whole plant of hornstedtia bella Škorničk
2020-01-01 Donadu, M. G.; Le, N. T.; Ho, D. V.; Doan, T. Q.; Le, A. T.; Raal, A.; Usai, M.; Marchetti, M.; Sanna, G.; Madeddu, S.; Rappelli, P.; Diaz, N.; Molicotti, P.; Carta, A.; Piras, S.; Usai, D.; Nguyen, H. T.; Cappuccinelli, P.; Zanetti, S.
Antiviral activity of benzotriazole based derivatives
2020-01-01 Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A.
Antiviral effect of Hornstedtia bella Škorničk essential oil from the whole plant against vaccinia virus (VV
2020-01-01 Sanna, Giuseppina; Madeddu, Silvia; Serreli, Gabriele; Thi Nguyen, Hoai; Trong Le, Nhan; Usai, Donatella; Carta, Antonio; Cappuccinelli, Piero; Zanetti &, Stefania; Gavino Donadu, Matthew
Biological activities of essential oils from leaves of paramignya trimera (Oliv.) guillaum and limnocitrus littoralis (miq.) swingle
2020-01-01 Le, N. T.; Ho, D. V.; Doan, T. Q.; Le, A. T.; Raal, A.; Usai, D.; Sanna, G.; Carta, A.; Rappelli, P.; Diaz, N.; Cappuccinelli, P.; Zanetti, S.; Nguyen, H. T.; Donadu, M. G.
Solid Lipid Nanoparticles as Formulative Strategy to Increase Oral Permeation of a Molecule Active in Multidrug-Resistant Tuberculosis Management
2020-01-01 Obinu, Antonella; Porcu, Elena Piera; Piras, Sandra; Ibba, Roberta; Carta, Antonio; Molicotti, Paola; Migheli, Rossana; Dalpiaz, Alessandro; Ferraro, Luca; Rassu, Giovanna; Gavini, Elisabetta; Giunchedi, Paolo
Anti-BVDV Activity Evaluation of Naphthoimidazole Derivatives Compared with Parental Imidazoquinoline Compounds
2020-01-01 Ibba, Roberta; Piras, Sandra; Delogu, Ilenia; Loddo, Roberta; Carta, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design, Synthesis, and Antiviral Activities of New Benzotriazole-Based Derivatives | 1-gen-2023 | Ibba, Roberta; Corona, Paola; Nonne, Francesca; Caria, Paola; Serreli, Gabriele; Palmas, Vanessa; Riu, Federico; Sestito, Simona; Nieddu, Maria; Loddo, Roberta; Sanna, Giuseppina; Piras, Sandra; Carta, Antonio | |
Improving in vivo oral bioavailability of a poorly soluble drug: a case study on polymeric versus lipid nanoparticles | 1-gen-2023 | Rassu, Giovanna; Obinu, Antonella; Serri, Carla; Piras, Sandra; Carta, Antonio; Ferraro, Luca; Gavini, Elisabetta; Giunchedi, Paolo; Dalpiaz, Alessandro | |
Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication | 1-gen-2022 | Ibba, Roberta; Riu, Federico; Delogu, Ilenia; Lupinu, Ilenia; Carboni, Gavino; Loddo, Roberta; Piras, Sandra; Carta, Antonio | |
A Lead-Based Fragment Library Screening of the Glycosyltransferase WaaG from Escherichia coli | 1-gen-2022 | Riu, Federico; Ruda, Alessandro; Engström, Olof; Muheim, Claudio; Mobarak, Hani; Ståhle, Jonas; Kosma, Paul; Carta, Antonio; Daley, Daniel O; Widmalm, Göran | |
Quinoxaline-based efflux pump inhibitors restore drug susceptibility in drug-resistant nontuberculous mycobacteria | 1-gen-2022 | Corona, Paola; Ibba, Roberta; Piras, Sandra; Molicotti, Paola; Bua, Alessandra; Carta, Antonio | |
Design, synthesis, and biological screening of a series of 4 '-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs) | 1-gen-2022 | Riu, F; Ibba, R; Zoroddu, S; Sestito, S; Lai, M; Piras, S; Sanna, L; Bordoni, V; Bagella, L; Carta, A | |
Design, synthesis, and biological screening of a series of 4′-fluoro-benzotriazole-acrylonitrile derivatives as microtubule-destabilising agents (MDAs) | 1-gen-2022 | Riu, Federico; Ibba, Roberta; Zoroddu, Stefano; Sestito, Simona; Lai, Michele; Piras, Sandra; Sanna, Luca; Bordoni, Valentina; Bagella, Luigi Marco; Carta, Antonio | |
Antibiotics and Carbohydrate-Containing Drugs Targeting Bacterial Cell Envelopes: An Overview | 1-gen-2022 | Riu, Federico; Ruda, Alessandro; Ibba, Roberta; Sestito, Simona; Lupinu, Ilenia; Piras, Sandra; Widmalm, Göran; Carta, Antonio | |
Human Enterovirus B: Selective Inhibition by Quinoxaline Derivatives and Bioinformatic RNA-Motif Identification as New Targets | 1-gen-2022 | Madeddu, Silvia; Ibba, Roberta; Sanna, Giuseppina; Piras, Sandra; Riu, Federico; Marongiu, Alessandra; Ambrosino, Annalisa; Caria, Paola; Onnis, Valentina; Franci, Gianluigi; Manzin, Aldo; Carta, Antonio | |
Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives | 1-gen-2021 | Ibba, R.; Piras, S.; Corona, P.; Riu, F.; Loddo, R.; Delogu, I.; Collu, G.; Sanna, G.; Caria, P.; Dettori, T.; Carta, A. | |
Inhibition of Enterovirus A71 by a Novel 2-Phenyl-Benzimidazole Derivative | 1-gen-2021 | Ibba, R.; Carta, A.; Madeddu, S.; Caria, P.; Serreli, G.; Piras, S.; Sestito, S.; Loddo, R.; Sanna, G. | |
A comprehensive assessment of a new series of 5′,6′-difluorobenzotriazole-acrylonitrile derivatives as microtubule targeting agents (MTAs) | 1-gen-2021 | Riu, F.; Sanna, L.; Ibba, R.; Piras, S.; Bordoni, V.; Scorciapino, M. A.; Lai, M.; Sestito, S.; Bagella, L.; Carta, A. | |
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. . | 1-gen-2021 | Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime | |
anti-BVDV Activity evaluation of Naphthoimidazole derivatives compared with parentalimidazoquinoline compounds | 1-gen-2020 | Ibba, Roberta; Piras, Sandra; Delogu, Ilenia; Loddo, Roberta; Carta, Antonio | |
Phytochemical compositions and biological activities of essential oils from the leaves, rhizomes and whole plant of hornstedtia bella Škorničk | 1-gen-2020 | Donadu, M. G.; Le, N. T.; Ho, D. V.; Doan, T. Q.; Le, A. T.; Raal, A.; Usai, M.; Marchetti, M.; Sanna, G.; Madeddu, S.; Rappelli, P.; Diaz, N.; Molicotti, P.; Carta, A.; Piras, S.; Usai, D.; Nguyen, H. T.; Cappuccinelli, P.; Zanetti, S. | |
Antiviral activity of benzotriazole based derivatives | 1-gen-2020 | Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A. | |
Antiviral effect of Hornstedtia bella Škorničk essential oil from the whole plant against vaccinia virus (VV | 1-gen-2020 | Sanna, Giuseppina; Madeddu, Silvia; Serreli, Gabriele; Thi Nguyen, Hoai; Trong Le, Nhan; Usai, Donatella; Carta, Antonio; Cappuccinelli, Piero; Zanetti &, Stefania; Gavino Donadu, Matthew | |
Biological activities of essential oils from leaves of paramignya trimera (Oliv.) guillaum and limnocitrus littoralis (miq.) swingle | 1-gen-2020 | Le, N. T.; Ho, D. V.; Doan, T. Q.; Le, A. T.; Raal, A.; Usai, D.; Sanna, G.; Carta, A.; Rappelli, P.; Diaz, N.; Cappuccinelli, P.; Zanetti, S.; Nguyen, H. T.; Donadu, M. G. | |
Solid Lipid Nanoparticles as Formulative Strategy to Increase Oral Permeation of a Molecule Active in Multidrug-Resistant Tuberculosis Management | 1-gen-2020 | Obinu, Antonella; Porcu, Elena Piera; Piras, Sandra; Ibba, Roberta; Carta, Antonio; Molicotti, Paola; Migheli, Rossana; Dalpiaz, Alessandro; Ferraro, Luca; Rassu, Giovanna; Gavini, Elisabetta; Giunchedi, Paolo | |
Anti-BVDV Activity Evaluation of Naphthoimidazole Derivatives Compared with Parental Imidazoquinoline Compounds | 1-gen-2020 | Ibba, Roberta; Piras, Sandra; Delogu, Ilenia; Loddo, Roberta; Carta, Antonio |
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