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RNAseq Analysis of Novel 1,3,4-Oxadiazole Chalcogen Analogues Reveals Anti-Tubulin Properties on Cancer Cell Lines 1-gen-2023 Zoroddu, Stefano; Sanna, Luca; Bordoni, Valentina; Lyu, Weidong; Murineddu, Gabriele; Pinna, Gerard A; Forcales, Sonia Vanina; Sala, Arturo; Kelvin, David J; Bagella, Luigi
Novel 1,3,4-oxadiazole chalcogen analogues: Synthesis and cytotoxic activity 1-gen-2022 Zoroddu, S.; Corona, P.; Sanna, L.; Borghi, F.; Bordoni, V.; Asproni, B.; Pinna, G. A.; Bagella, L.; Murineddu, G.
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction 1-gen-2021 Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A.
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. . 1-gen-2021 Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime
Chimica farmaceutica. Con e-book 1-gen-2020 Pinna, Gerard; Murineddu, Gabriele
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes 1-gen-2020 Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A.
Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties 1-gen-2020 Weidong, L.; Sanna, L.; Bordoni, V.; Tiansheng, Z.; Chengxun, L.; Murineddu, G.; Pinna, G. A.; Kelvin, D. J.; Bagella, L.
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation 1-gen-2019 Asproni, Battistina; Murineddu, Gabriele; Lazzari, Paolo; Pinna, Gerard A.
A diethylpyrocarbonate-based derivatization method for the LC-MS/MS measurement of plasma arginine and its chemically related metabolites and analogs 1-gen-2019 Sotgia, Salvatore; Zinellu, Angelo; Paliogiannis, Panagiotis; Pinna, Gerard A.; Mangoni, Arduino A.; Milanesi, Luciano; Carru, Ciriaco
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors 1-gen-2019 Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A.
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands 1-gen-2019 Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A.
Hercynine content in widely consumed commercial beverages 1-gen-2018 Sotgia, Salvatore; Zinellu, Angelo; Forteschi, Mauro; Paliogiannis, Panagiotis; Pinna, Gerard A.; Mangoni, Arduino A.; Carru, Ciriaco
A liquid chromatography-mass spectrometry study on the spirocyclization of ninhydrin with the aminothiols 1-gen-2018 Sotgia, Salvatore; Zinellu, Angelo; Forteschi, Mauro; Paliogiannis, Panagiotis; Deiana, Giovanni A.; Pinna, Gerard A.; Mangoni, Arduino A.; Carru, Ciriaco
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands 1-gen-2018 Asproni, B.; Manca, I.; Pinna, G.; Cichero, E.; Fossa, P.; Murineddu, G.; Lazzari, P.; Loriga, Maria Giovanna; Pinna, G. A
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists 1-gen-2018 Murineddu, Gabriele; Deligia, Francesco; Ragusa, Giulio; García-Toscano, Laura; Gómez-Cañas, María; Asproni, Battistina; Satta, Valentina; Cichero, Elena; Pazos, Ruth; Fossa, Paola; Loriga, Giovanni; Fernández-Ruiz, Javier; Pinna, Gerard A.
Development of an LC-Tandem Mass Spectrometry Method for the Quantitative Analysis of Hercynine in Human Whole Blood 1-gen-2018 Sotgia, Salvatore; Murphy, Rhys B.; Zinellu, Angelo; Elliot, David; Paliogiannis, Panagiotis; Pinna, Gerard Aime; Carru, Ciriaco; Mangoni, Arduino A.
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands 1-gen-2018 Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS 1-gen-2018 Deligia, Francesco; Murineddu, Gabriele; Cecilia, Gotti; Ragusa, Giulio; Francesca, Fasoli; Miriam, Sciaccaluga; Simona, Plutino; Sergio, Fucile; Giovanni, Loriga; Asproni, Battistina; Pinna, Gerard A.
I farmaci antivirali. Dalla progettazione all’impiego terapeutico. 1-gen-2017 Carta, A.; Murineddu, G.; Pinna, G. A.
New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking 1-gen-2017 Ragusa, Giulio; Gomez Cañas, M.; Morales, P.; Rodríguez Cueto, C.; Pazos, M. R.; Asproni, Battistina; Cichero, E.; Fossa, P.; Pinna, Gerard Aime; Jagerovic, N.; Fernandez Ruiz, J.; Murineddu, Gabriele
Mostrati risultati da 1 a 20 di 275
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