Sfoglia per Autore
Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction
2023-01-01 Asproni, Battistina; Catto, Marco; Loriga, Giovanni; Murineddu, Gabriele; Corona, Paola; Purgatorio, Rosa; Cichero, Elena; Fossa, Paola; Scarano, Naomi; Martínez, Anto ́n L.; ́e Brea, Jos; Pinna, G ́erard A.
RNAseq Analysis of Novel 1,3,4-Oxadiazole Chalcogen Analogues Reveals Anti-Tubulin Properties on Cancer Cell Lines
2023-01-01 Zoroddu, Stefano; Sanna, Luca; Bordoni, Valentina; Lyu, Weidong; Murineddu, Gabriele; Pinna, Gerard A; Forcales, Sonia Vanina; Sala, Arturo; Kelvin, David J; Bagella, Luigi
Novel 1,3,4-oxadiazole chalcogen analogues: Synthesis and cytotoxic activity
2022-01-01 Zoroddu, S.; Corona, P.; Sanna, L.; Borghi, F.; Bordoni, V.; Asproni, B.; Pinna, G. A.; Bagella, L.; Murineddu, G.
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. .
2021-01-01 Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction
2021-01-01 Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A.
Chimica farmaceutica. Con e-book
2020-01-01 Pinna, Gerard; Murineddu, Gabriele
Antiviral activity of benzotriazole based derivatives
2020-01-01 Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A.
Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties
2020-01-01 Weidong, L.; Sanna, L.; Bordoni, V.; Tiansheng, Z.; Chengxun, L.; Murineddu, G.; Pinna, G. A.; Kelvin, D. J.; Bagella, L.
Preliminary anti-coxsackie activity of novel 1-[4-(5,6-dimethyl(h)1h(2h)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas
2020-01-01 Piras, S.; Corona, P.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A.
Antiviral Activity of Benzotriazole Based Derivatives
2020-01-01 Corona, Paola; Piras, Sandra; Ibba, Roberta; Riu, Federico; Murineddu, Gabriele; Sanna, Giuseppina; Madeddu, Silvia; Delogu, Ilenia; Loddo and Antonio Carta, Roberta
5,6-Dichloro-2-phenyl-benzotriazoles: New potent inhibitors of orthohantavirus
2020-01-01 Sanna, G.; Piras, S.; Madeddu, S.; Busonera, B.; Klempa, B.; Corona, P.; Ibba, R.; Murineddu, G.; Carta, A.; Loddo, R.
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes
2020-01-01 Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A.
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation
2019-01-01 Asproni, Battistina; Murineddu, Gabriele; Lazzari, Paolo; Pinna, Gerard A.
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors
2019-01-01 Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A.
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands
2019-01-01 Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A.
Principi generali. In: Chimica Tossicologica
2018-01-01 Murineddu, G
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists
2018-01-01 Murineddu, Gabriele; Deligia, Francesco; Ragusa, Giulio; García-Toscano, Laura; Gómez-Cañas, María; Asproni, Battistina; Satta, Valentina; Cichero, Elena; Pazos, Ruth; Fossa, Paola; Loriga, Giovanni; Fernández-Ruiz, Javier; Pinna, Gerard A.
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands
2018-01-01 Asproni, B.; Manca, I.; Pinna, G.; Cichero, E.; Fossa, P.; Murineddu, G.; Lazzari, P.; Loriga, Maria Giovanna; Pinna, G. A
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS
2018-01-01 Deligia, Francesco; Murineddu, Gabriele; Cecilia, Gotti; Ragusa, Giulio; Francesca, Fasoli; Miriam, Sciaccaluga; Simona, Plutino; Sergio, Fucile; Giovanni, Loriga; Asproni, Battistina; Pinna, Gerard A.
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands
2018-01-01 Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction | 1-gen-2023 | Asproni, Battistina; Catto, Marco; Loriga, Giovanni; Murineddu, Gabriele; Corona, Paola; Purgatorio, Rosa; Cichero, Elena; Fossa, Paola; Scarano, Naomi; Martínez, Anto ́n L.; ́e Brea, Jos; Pinna, G ́erard A. | |
RNAseq Analysis of Novel 1,3,4-Oxadiazole Chalcogen Analogues Reveals Anti-Tubulin Properties on Cancer Cell Lines | 1-gen-2023 | Zoroddu, Stefano; Sanna, Luca; Bordoni, Valentina; Lyu, Weidong; Murineddu, Gabriele; Pinna, Gerard A; Forcales, Sonia Vanina; Sala, Arturo; Kelvin, David J; Bagella, Luigi | |
Novel 1,3,4-oxadiazole chalcogen analogues: Synthesis and cytotoxic activity | 1-gen-2022 | Zoroddu, S.; Corona, P.; Sanna, L.; Borghi, F.; Bordoni, V.; Asproni, B.; Pinna, G. A.; Bagella, L.; Murineddu, G. | |
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. . | 1-gen-2021 | Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime | |
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction | 1-gen-2021 | Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A. | |
Chimica farmaceutica. Con e-book | 1-gen-2020 | Pinna, Gerard; Murineddu, Gabriele | |
Antiviral activity of benzotriazole based derivatives | 1-gen-2020 | Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A. | |
Target identification of a novel unsymmetrical 1,3,4-oxadiazole derivative with antiproliferative properties | 1-gen-2020 | Weidong, L.; Sanna, L.; Bordoni, V.; Tiansheng, Z.; Chengxun, L.; Murineddu, G.; Pinna, G. A.; Kelvin, D. J.; Bagella, L. | |
Preliminary anti-coxsackie activity of novel 1-[4-(5,6-dimethyl(h)1h(2h)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas | 1-gen-2020 | Piras, S.; Corona, P.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A. | |
Antiviral Activity of Benzotriazole Based Derivatives | 1-gen-2020 | Corona, Paola; Piras, Sandra; Ibba, Roberta; Riu, Federico; Murineddu, Gabriele; Sanna, Giuseppina; Madeddu, Silvia; Delogu, Ilenia; Loddo and Antonio Carta, Roberta | |
5,6-Dichloro-2-phenyl-benzotriazoles: New potent inhibitors of orthohantavirus | 1-gen-2020 | Sanna, G.; Piras, S.; Madeddu, S.; Busonera, B.; Klempa, B.; Corona, P.; Ibba, R.; Murineddu, G.; Carta, A.; Loddo, R. | |
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes | 1-gen-2020 | Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A. | |
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation | 1-gen-2019 | Asproni, Battistina; Murineddu, Gabriele; Lazzari, Paolo; Pinna, Gerard A. | |
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors | 1-gen-2019 | Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A. | |
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands | 1-gen-2019 | Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A. | |
Principi generali. In: Chimica Tossicologica | 1-gen-2018 | Murineddu, G | |
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists | 1-gen-2018 | Murineddu, Gabriele; Deligia, Francesco; Ragusa, Giulio; García-Toscano, Laura; Gómez-Cañas, María; Asproni, Battistina; Satta, Valentina; Cichero, Elena; Pazos, Ruth; Fossa, Paola; Loriga, Giovanni; Fernández-Ruiz, Javier; Pinna, Gerard A. | |
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands | 1-gen-2018 | Asproni, B.; Manca, I.; Pinna, G.; Cichero, E.; Fossa, P.; Murineddu, G.; Lazzari, P.; Loriga, Maria Giovanna; Pinna, G. A | |
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS | 1-gen-2018 | Deligia, Francesco; Murineddu, Gabriele; Cecilia, Gotti; Ragusa, Giulio; Francesca, Fasoli; Miriam, Sciaccaluga; Simona, Plutino; Sergio, Fucile; Giovanni, Loriga; Asproni, Battistina; Pinna, Gerard A. | |
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands | 1-gen-2018 | Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile