Sfoglia per Autore
Integrase
2023-01-01 Carta, Fabrizio; Sechi, Mario
α-Glucosidase inhibition by green, white and oolong teas: in vitro activity and computational studies
2023-01-01 Esposito, Fabio; Pala, Nicolino; Carcelli, Mauro; Boateng, Samuel T; D'Aquila, Paolo S; Mariani, Alberto; Satta, Sandro; Chamcheu, Jean Christopher; Sechi, Mario; Sanna, Vanna
Synthesis, in silico modelling, and in vitro biological evaluation of substituted pyrazole derivatives as potential anti-skin cancer, anti-tyrosinase, and antioxidant agents
2023-01-01 Boateng, Samuel T.; Roy, Tithi; Torrey, Kara; Owunna, Uchechi; Banang-Mbeumi, Sergette; Basnet, David; Niedda, Eleonora; Alexander, Alexis D.; Hage, Denzel El; Atchimnaidu, Siriki; Nagalo, Bolni Marius; Aryal, Dinesh; Findley, Ann; Seeram, Navindra P.; Efimova, Tatiana; Sechi, Mario; Hill, Ronald A.; Ma, Hang; Chamcheu, Jean Christopher; Murru, Siva
Comparative efficacy of epigallocatechin gallate and its nano-formulation in prostate cancer 3D spheroids model
2023-01-01 Alserihi, Read F.; Mohammed, Mohammed Razeeth Shait; Kaleem, Mohammed; Imran Khan, Mohammad; Sechi, Mario; Zughaibi, Torki A.; Tabrez, Shams
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches
2022-01-01 Pagnozzi, Daniela; Pala, Nicolino; Biosa, Grazia; Dallocchio, Roberto Nico; Dess??, Alessandro; Singh, Pankaj Kumar; Rogolino, Dominga; Di Fiore, Anna; De Simone, Giuseppina; Supuran, Claudiu T.; Sechi, Mario
Development of targeted nanoparticles loaded with antiviral drugs for SARS-CoV-2 inhibition
2022-01-01 Sanna, Vanna Annunziata; Satta, Sandro; Hsiai, Tzung; Sechi, Mario
Development of Targeted Nanoparticles Loaded with Antiviral Drugs for SARS-CoV-2 Inhibition
2021-01-01 Sanna, Vanna; Satta, Sandro; Hsiai, Tzung; Sechi, Mario
Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers
2021-01-01 Roy, Tithi; Boateng, Samuel T.; Banang-Mbeumi, Sergette; Singh, Pankaj K.; Basnet, Pratik; Chamcheu, Roxane-Cherille N.; Ladu, Federico; Chauvin, Isabel; Spiegelman, Vladimir S.; Hill, Ronald A.; Kousoulas, Konstantin G.; Nagalo, Bolni Marius; Walker, Anthony L.; Fotie, Jean; Murru, Siva; Sechi, Mario; Chamcheu, Jean Christopher
Identification of new fisetin analogs as kinase inhibitors: Data on synthesis and anti-skin cancer activities evaluation
2021-01-01 Roy, Tithi; Boateng, Samuel T; Banang-Mbeumi, Sergette; Singh, Pankaj K; Basnet, Pratik; Chamcheu, Roxane-Cherille N; Ladu, Federico; Chauvin, Isabel; Spiegelman, Vladimir S; Hill, Ronald A; Kousoulas, Konstantin G; Nagalo, Bolni Marius; Walker, Anthony L; Fotie, Jean; Murru, Siva; Sechi, Mario; Chamcheu, Jean Christopher
Development of (-)-epigallocatechin-3-gallate-loaded folate receptor-targeted nanoparticles for prostate cancer treatment
2021-01-01 Alserihi, Read F.; Razeeth Shait Mohammed, Mohammed; Kaleem, Mohammed; Imran Khan, Mohammad; Sechi, Mario; Sanna, Vanna Annunziata; Zughaibi, Torki A.; Abuzenadah, Adel M.; Tabrez, Shams
Inhibition of Human Immunodeficiency Virus-1 Integrase by β-Diketo Acid Coated Gold Nanoparticles
2020-01-01 Sanna, V.; Youssef, M. F.; Pala, N.; Rogolino, D.; Carcelli, M.; Singh, P. K.; Sanchez, T.; Neamati, N.; Sechi, M.
Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitors
2020-01-01 Esposito, F.; Sechi, M.; Pala, N.; Sanna, A.; Koneru, P. C.; Kvaratskhelia, M.; Naesens, L.; Corona, A.; Grandi, N.; di Santo, R.; D'Amore, V. M.; Di Leva, F. S.; Novellino, E.; Cosconati, S.; Tramontano, E.
A Novel Redox Modulator Induces a GPX4-Mediated Cell Death That Is Dependent on Iron and Reactive Oxygen Species
2020-01-01 Hu, S.; Sechi, M.; Singh, P. K.; Dai, L.; Mccann, S.; Sun, D.; Ljungman, M.; Neamati, N.
Diketo acids inhibit the cap-snatching endonuclease of several Bunyavirales
2020-01-01 Fernandez-Garcia, Y.; Horst, S. T.; Bassetto, M.; Brancale, A.; Neyts, J.; Rogolino, D.; Sechi, M.; Carcelli, M.; Gunther, S.; Rocha-Pereira, J.
Therapeutic Potential of Targeted Nanoparticles and Perspective on Nanotherapies
2020-01-01 Sanna, V.; Sechi, M.
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture
2020-01-01 Pala, N.; Esposito, F.; Tramontano, E.; Singh, P. K.; Sanna, V.; Carcelli, M.; Haigh, L. D.; Satta, S.; Sechi, M.
Discovery of novel functionalized 1,2,4-triazoles as PARP-1 inhibitors in breast cancer: Design, synthesis and antitumor activity evaluation
2019-01-01 Boraei, A. T. A.; Singh, Pankaj Kumar; Sechi, M.; Satta, Sandro
Proproliferative function of adaptor protein GRB10 in prostate carcinoma
2019-01-01 Khan, Mohammad Imran; Al Johani, Ahmed; Hamid, Abid; Ateeq, Bushra; Manzar, Nishat; Adhami, Vaqar Mustafa; Lall, Rahul K; Rath, Suvasmita; Sechi, Mario; Siddiqui, Imtiaz Ahmad; Choudhry, Hani; Zamzami, Mazin A; Havighurst, Thomas C; Huang, Wei; Ntambi, James M; Mukhtar, Hasan
Fisetin targets YB-1/RSK axis independent of its effect on ERK signaling: insights from in vitro and in vivo melanoma models
2018-01-01 Sechi, Mario; Lall, Rahul K.; Afolabi, Saheed O; Singh, Anant; Joshi, Dinesh C.; Chiu, Shing-Yan; Mukhtar, Hasan; Syed, Deeba N.
Design and Synthesis of Novel Reactive Oxygen Species Inducers for the Treatment of Pancreatic Ductal Adenocarcinoma
2018-01-01 Kuang, Yuting; Sechi, Mario; Nurra, Salvatore; Ljungman, Mats; Neamati, Nouri
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Integrase | 1-gen-2023 | Carta, Fabrizio; Sechi, Mario | |
α-Glucosidase inhibition by green, white and oolong teas: in vitro activity and computational studies | 1-gen-2023 | Esposito, Fabio; Pala, Nicolino; Carcelli, Mauro; Boateng, Samuel T; D'Aquila, Paolo S; Mariani, Alberto; Satta, Sandro; Chamcheu, Jean Christopher; Sechi, Mario; Sanna, Vanna | |
Synthesis, in silico modelling, and in vitro biological evaluation of substituted pyrazole derivatives as potential anti-skin cancer, anti-tyrosinase, and antioxidant agents | 1-gen-2023 | Boateng, Samuel T.; Roy, Tithi; Torrey, Kara; Owunna, Uchechi; Banang-Mbeumi, Sergette; Basnet, David; Niedda, Eleonora; Alexander, Alexis D.; Hage, Denzel El; Atchimnaidu, Siriki; Nagalo, Bolni Marius; Aryal, Dinesh; Findley, Ann; Seeram, Navindra P.; Efimova, Tatiana; Sechi, Mario; Hill, Ronald A.; Ma, Hang; Chamcheu, Jean Christopher; Murru, Siva | |
Comparative efficacy of epigallocatechin gallate and its nano-formulation in prostate cancer 3D spheroids model | 1-gen-2023 | Alserihi, Read F.; Mohammed, Mohammed Razeeth Shait; Kaleem, Mohammed; Imran Khan, Mohammad; Sechi, Mario; Zughaibi, Torki A.; Tabrez, Shams | |
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches | 1-gen-2022 | Pagnozzi, Daniela; Pala, Nicolino; Biosa, Grazia; Dallocchio, Roberto Nico; Dess??, Alessandro; Singh, Pankaj Kumar; Rogolino, Dominga; Di Fiore, Anna; De Simone, Giuseppina; Supuran, Claudiu T.; Sechi, Mario | |
Development of targeted nanoparticles loaded with antiviral drugs for SARS-CoV-2 inhibition | 1-gen-2022 | Sanna, Vanna Annunziata; Satta, Sandro; Hsiai, Tzung; Sechi, Mario | |
Development of Targeted Nanoparticles Loaded with Antiviral Drugs for SARS-CoV-2 Inhibition | 1-gen-2021 | Sanna, Vanna; Satta, Sandro; Hsiai, Tzung; Sechi, Mario | |
Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers | 1-gen-2021 | Roy, Tithi; Boateng, Samuel T.; Banang-Mbeumi, Sergette; Singh, Pankaj K.; Basnet, Pratik; Chamcheu, Roxane-Cherille N.; Ladu, Federico; Chauvin, Isabel; Spiegelman, Vladimir S.; Hill, Ronald A.; Kousoulas, Konstantin G.; Nagalo, Bolni Marius; Walker, Anthony L.; Fotie, Jean; Murru, Siva; Sechi, Mario; Chamcheu, Jean Christopher | |
Identification of new fisetin analogs as kinase inhibitors: Data on synthesis and anti-skin cancer activities evaluation | 1-gen-2021 | Roy, Tithi; Boateng, Samuel T; Banang-Mbeumi, Sergette; Singh, Pankaj K; Basnet, Pratik; Chamcheu, Roxane-Cherille N; Ladu, Federico; Chauvin, Isabel; Spiegelman, Vladimir S; Hill, Ronald A; Kousoulas, Konstantin G; Nagalo, Bolni Marius; Walker, Anthony L; Fotie, Jean; Murru, Siva; Sechi, Mario; Chamcheu, Jean Christopher | |
Development of (-)-epigallocatechin-3-gallate-loaded folate receptor-targeted nanoparticles for prostate cancer treatment | 1-gen-2021 | Alserihi, Read F.; Razeeth Shait Mohammed, Mohammed; Kaleem, Mohammed; Imran Khan, Mohammad; Sechi, Mario; Sanna, Vanna Annunziata; Zughaibi, Torki A.; Abuzenadah, Adel M.; Tabrez, Shams | |
Inhibition of Human Immunodeficiency Virus-1 Integrase by β-Diketo Acid Coated Gold Nanoparticles | 1-gen-2020 | Sanna, V.; Youssef, M. F.; Pala, N.; Rogolino, D.; Carcelli, M.; Singh, P. K.; Sanchez, T.; Neamati, N.; Sechi, M. | |
Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitors | 1-gen-2020 | Esposito, F.; Sechi, M.; Pala, N.; Sanna, A.; Koneru, P. C.; Kvaratskhelia, M.; Naesens, L.; Corona, A.; Grandi, N.; di Santo, R.; D'Amore, V. M.; Di Leva, F. S.; Novellino, E.; Cosconati, S.; Tramontano, E. | |
A Novel Redox Modulator Induces a GPX4-Mediated Cell Death That Is Dependent on Iron and Reactive Oxygen Species | 1-gen-2020 | Hu, S.; Sechi, M.; Singh, P. K.; Dai, L.; Mccann, S.; Sun, D.; Ljungman, M.; Neamati, N. | |
Diketo acids inhibit the cap-snatching endonuclease of several Bunyavirales | 1-gen-2020 | Fernandez-Garcia, Y.; Horst, S. T.; Bassetto, M.; Brancale, A.; Neyts, J.; Rogolino, D.; Sechi, M.; Carcelli, M.; Gunther, S.; Rocha-Pereira, J. | |
Therapeutic Potential of Targeted Nanoparticles and Perspective on Nanotherapies | 1-gen-2020 | Sanna, V.; Sechi, M. | |
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture | 1-gen-2020 | Pala, N.; Esposito, F.; Tramontano, E.; Singh, P. K.; Sanna, V.; Carcelli, M.; Haigh, L. D.; Satta, S.; Sechi, M. | |
Discovery of novel functionalized 1,2,4-triazoles as PARP-1 inhibitors in breast cancer: Design, synthesis and antitumor activity evaluation | 1-gen-2019 | Boraei, A. T. A.; Singh, Pankaj Kumar; Sechi, M.; Satta, Sandro | |
Proproliferative function of adaptor protein GRB10 in prostate carcinoma | 1-gen-2019 | Khan, Mohammad Imran; Al Johani, Ahmed; Hamid, Abid; Ateeq, Bushra; Manzar, Nishat; Adhami, Vaqar Mustafa; Lall, Rahul K; Rath, Suvasmita; Sechi, Mario; Siddiqui, Imtiaz Ahmad; Choudhry, Hani; Zamzami, Mazin A; Havighurst, Thomas C; Huang, Wei; Ntambi, James M; Mukhtar, Hasan | |
Fisetin targets YB-1/RSK axis independent of its effect on ERK signaling: insights from in vitro and in vivo melanoma models | 1-gen-2018 | Sechi, Mario; Lall, Rahul K.; Afolabi, Saheed O; Singh, Anant; Joshi, Dinesh C.; Chiu, Shing-Yan; Mukhtar, Hasan; Syed, Deeba N. | |
Design and Synthesis of Novel Reactive Oxygen Species Inducers for the Treatment of Pancreatic Ductal Adenocarcinoma | 1-gen-2018 | Kuang, Yuting; Sechi, Mario; Nurra, Salvatore; Ljungman, Mats; Neamati, Nouri |
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