Sfoglia per Autore
Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction
2023-01-01 Asproni, Battistina; Catto, Marco; Loriga, Giovanni; Murineddu, Gabriele; Corona, Paola; Purgatorio, Rosa; Cichero, Elena; Fossa, Paola; Scarano, Naomi; Martínez, Anto ́n L.; ́e Brea, Jos; Pinna, G ́erard A.
Novel 1,3,4-oxadiazole chalcogen analogues: Synthesis and cytotoxic activity
2022-01-01 Zoroddu, S.; Corona, P.; Sanna, L.; Borghi, F.; Bordoni, V.; Asproni, B.; Pinna, G. A.; Bagella, L.; Murineddu, G.
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction
2021-01-01 Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A.
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. .
2021-01-01 Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes
2020-01-01 Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A.
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation
2019-01-01 Asproni, Battistina; Murineddu, Gabriele; Lazzari, Paolo; Pinna, Gerard A.
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands
2019-01-01 Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A.
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors
2019-01-01 Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A.
Biotrasformazione degli xenobiotici. In: Chimica Tossicologica
2018-01-01 Asproni, Battistina
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS
2018-01-01 Deligia, Francesco; Murineddu, Gabriele; Cecilia, Gotti; Ragusa, Giulio; Francesca, Fasoli; Miriam, Sciaccaluga; Simona, Plutino; Sergio, Fucile; Giovanni, Loriga; Asproni, Battistina; Pinna, Gerard A.
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists
2018-01-01 Murineddu, Gabriele; Deligia, Francesco; Ragusa, Giulio; García-Toscano, Laura; Gómez-Cañas, María; Asproni, Battistina; Satta, Valentina; Cichero, Elena; Pazos, Ruth; Fossa, Paola; Loriga, Giovanni; Fernández-Ruiz, Javier; Pinna, Gerard A.
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands
2018-01-01 Asproni, B.; Manca, I.; Pinna, G.; Cichero, E.; Fossa, P.; Murineddu, G.; Lazzari, P.; Loriga, Maria Giovanna; Pinna, G. A
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands
2018-01-01 Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele
Correction to Synthesis and antineoplastic evaluation of novel unsymmetrical 1,3,4-oxadiazoles
2017-01-01 Nieddu, Valentina; Pinna, Giansalvo; Marchesi, Irene; Sanna, Luca; Asproni, Battistina; Pinna, Gerard Aime; Bagella, L.; Murineddu, Gabriele
New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking
2017-01-01 Ragusa, Giulio; Gomez Cañas, M.; Morales, P.; Rodríguez Cueto, C.; Pazos, M. R.; Asproni, Battistina; Cichero, E.; Fossa, P.; Pinna, Gerard Aime; Jagerovic, N.; Fernandez Ruiz, J.; Murineddu, Gabriele
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism
2016-01-01 Fois, G. R.; Fattore, L.; Murineddu, Gabriele; Salis, A.; Pintore, Giorgio Antonio Mario; Asproni, Battistina; Pinna, Gerard Aime; Diana, Marco
Tricyclic Pyrazoles. Part 8. Synthesis, Biological Evaluation and Modelling of Tricyclic Pyrazole Carboxamides as Potential CB2 Receptor Ligands with Antagonist/Inverse Agonist Properties.
2016-01-01 Deiana, V; Gómez Cañas, M; Pazos, M. R.; Fernández Ruiz, J; Asproni, B; Cichero, E; Fossa, P; Muñoz, E; Deligia, F; Murineddu, Gabriele; García Arencibia, M; Pinna, Gerard Aime
Synthesis and Antineoplastic Evaluation of Novel Unsymmetrical 1,3,4-Oxadiazoles
2016-01-01 Nieddu, Valentina; Pinna, Giansalvo; Marchesi, Irene; Sanna, Luca; Asproni, Battistina; Pinna, Gerard Aime; Bagella, Luigi Marco; Murineddu, Gabriele
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonists
2016-01-01 Dore, A.; Asproni, Battistina; Scampuddu, A.; Gessi, S.; Murineddu, Gabriele; Cichero, E.; Fossa, P.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime
Synthesis and binding affinity of N-6 biaryl-N-propionyl-3,6-diazabicyclo[3.1.1]heptanes.
2015-01-01 Pinna, Giov; Dore, A.; Asproni, B.; Pinna, Gians; Gessi, S.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT6 receptor interaction | 1-gen-2023 | Asproni, Battistina; Catto, Marco; Loriga, Giovanni; Murineddu, Gabriele; Corona, Paola; Purgatorio, Rosa; Cichero, Elena; Fossa, Paola; Scarano, Naomi; Martínez, Anto ́n L.; ́e Brea, Jos; Pinna, G ́erard A. | |
Novel 1,3,4-oxadiazole chalcogen analogues: Synthesis and cytotoxic activity | 1-gen-2022 | Zoroddu, S.; Corona, P.; Sanna, L.; Borghi, F.; Bordoni, V.; Asproni, B.; Pinna, G. A.; Bagella, L.; Murineddu, G. | |
Tricyclic Pyrazole-Based Compounds as Useful Scaffolds for Cannabinoid CB1/CB2 Receptor Interaction | 1-gen-2021 | Asproni, B.; Murineddu, G.; Corona, P.; Pinna, G. A. | |
Biological Effects on μ-Receptors Affinity and Selectivity of Arylpropenyl Chain Structural Modification on Diazatricyclodecane Derivatives. . | 1-gen-2021 | Piras, Sandra; Murineddu, Gabriele; Loriga2, Giovanni; Carta, Antonio; Battistello, Enrica; Merighi, Stefania; Gessi, Stefania; Corona, Paola; Asproni, Battistina; Ibba, Roberta; Temml, Veronika; Schuster, Daniela; Pinna, Gerard Aime | |
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes | 1-gen-2020 | Murineddu, G.; Asproni, B.; Corona, P.; Gessi, S.; Merighi, S.; Battistello, E.; Sturaro, C.; Calo, G.; Galeotti, N.; Temml, V.; Herdlinger, S.; Schuster, D.; Pinna, G. A. | |
Tricyclic thienopyrazole derivatives as ligands for cannabinoid receptors: synthesis and biological evaluation | 1-gen-2019 | Asproni, Battistina; Murineddu, Gabriele; Lazzari, Paolo; Pinna, Gerard A. | |
Development of oxygen-bridged pyrazole-based structures as cannabinoid receptor 1 ligands | 1-gen-2019 | Murineddu, Gabriele; Asproni, Battistina; Corona, Paola; Piras, Sandra; Lazzari, Paolo; Ruiu, Stefania; Legnani, Laura; Toma, Lucio; Pinna, Gerard A. | |
Novel N-aryl nicotinamide derivatives: tacking stock on 3,6-diazabicyclo[3.3.1]heptanes as ligands for neuronal acetylcholine receptors | 1-gen-2019 | Murineddu, G.; Gotti, C.; Asproni, B.; Corona, P.; Martinello, K.; Plutino, S.; Fucile, S.; Temml, V.; Moretti, M.; Viani, P.; Schuster, D.; Piras, S.; Deligia, F.; Pinna, G. A. | |
Biotrasformazione degli xenobiotici. In: Chimica Tossicologica | 1-gen-2018 | Asproni, Battistina | |
Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: novel selective ligands with subnanomolar affinity for α4β2 nACh receptorS | 1-gen-2018 | Deligia, Francesco; Murineddu, Gabriele; Cecilia, Gotti; Ragusa, Giulio; Francesca, Fasoli; Miriam, Sciaccaluga; Simona, Plutino; Sergio, Fucile; Giovanni, Loriga; Asproni, Battistina; Pinna, Gerard A. | |
Novel sulfenamides and sulfonamides based on pyridazinone and pyridazine scaffolds as CB1 receptor ligand antagonists | 1-gen-2018 | Murineddu, Gabriele; Deligia, Francesco; Ragusa, Giulio; García-Toscano, Laura; Gómez-Cañas, María; Asproni, Battistina; Satta, Valentina; Cichero, Elena; Pazos, Ruth; Fossa, Paola; Loriga, Giovanni; Fernández-Ruiz, Javier; Pinna, Gerard A. | |
Novel pyrrolocycloalkylpyrazole analogues as CB1 ligands | 1-gen-2018 | Asproni, B.; Manca, I.; Pinna, G.; Cichero, E.; Fossa, P.; Murineddu, G.; Lazzari, P.; Loriga, Maria Giovanna; Pinna, G. A | |
Synthesis, Pharmacological Evaluation, and Docking Studies of Novel Pyridazinone-Based Cannabinoid Receptor Type 2 Ligands | 1-gen-2018 | Ragusa, Giulio; Bencivenni, Serena; Morales, Paula; Callaway, Tyra; Hurst, Dr. Dow. P.; Asproni, Battistina; Merighi, Stefania; Loriga, Giovanni; Pinna, Gerard A.; Reggio, Patricia H.; Gessi, Stefania; Murineddu, Gabriele | |
Correction to Synthesis and antineoplastic evaluation of novel unsymmetrical 1,3,4-oxadiazoles | 1-gen-2017 | Nieddu, Valentina; Pinna, Giansalvo; Marchesi, Irene; Sanna, Luca; Asproni, Battistina; Pinna, Gerard Aime; Bagella, L.; Murineddu, Gabriele | |
New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking | 1-gen-2017 | Ragusa, Giulio; Gomez Cañas, M.; Morales, P.; Rodríguez Cueto, C.; Pazos, M. R.; Asproni, Battistina; Cichero, E.; Fossa, P.; Pinna, Gerard Aime; Jagerovic, N.; Fernandez Ruiz, J.; Murineddu, Gabriele | |
The novel cannabinoid antagonist SM-11 reduces hedonic aspect of food intake through a dopamine-dependent mechanism | 1-gen-2016 | Fois, G. R.; Fattore, L.; Murineddu, Gabriele; Salis, A.; Pintore, Giorgio Antonio Mario; Asproni, Battistina; Pinna, Gerard Aime; Diana, Marco | |
Tricyclic Pyrazoles. Part 8. Synthesis, Biological Evaluation and Modelling of Tricyclic Pyrazole Carboxamides as Potential CB2 Receptor Ligands with Antagonist/Inverse Agonist Properties. | 1-gen-2016 | Deiana, V; Gómez Cañas, M; Pazos, M. R.; Fernández Ruiz, J; Asproni, B; Cichero, E; Fossa, P; Muñoz, E; Deligia, F; Murineddu, Gabriele; García Arencibia, M; Pinna, Gerard Aime | |
Synthesis and Antineoplastic Evaluation of Novel Unsymmetrical 1,3,4-Oxadiazoles | 1-gen-2016 | Nieddu, Valentina; Pinna, Giansalvo; Marchesi, Irene; Sanna, Luca; Asproni, Battistina; Pinna, Gerard Aime; Bagella, Luigi Marco; Murineddu, Gabriele | |
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB2 receptor antagonists/inverse agonists | 1-gen-2016 | Dore, A.; Asproni, Battistina; Scampuddu, A.; Gessi, S.; Murineddu, Gabriele; Cichero, E.; Fossa, P.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime | |
Synthesis and binding affinity of N-6 biaryl-N-propionyl-3,6-diazabicyclo[3.1.1]heptanes. | 1-gen-2015 | Pinna, Giov; Dore, A.; Asproni, B.; Pinna, Gians; Gessi, S.; Merighi, S.; Bencivenni, S.; Pinna, Gerard Aime |
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